SCHEMBL17713670

SCHEMBL17713670

Cc1cc(C)c(CNC(=O)c2csc(CCCC3CCN(CC(C)(C)F)CC3)c2C)c(=O)[nH]1

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EED O75530 20/20 0.56
RBBP4 Q09028 20/20 0.56
SUZ12 Q15022 20/20 0.56
EZH2 Q15910 20/20 0.56
AEBP2 Q6ZN18 20/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17713687 0.95 EED (0.56) EEDRBBP4SUZ12EZH2AEBP2
SCHEMBL17713684 0.94 EZH2 (0.55) EEDRBBP4SUZ12EZH2AEBP2
SCHEMBL17713702 0.91 EED (0.55) EEDRBBP4SUZ12EZH2AEBP2
SCHEMBL17713650 0.89 EED (0.56) EEDRBBP4SUZ12EZH2AEBP2
SCHEMBL16212764 0.87 EED (0.60) EEDRBBP4SUZ12EZH2AEBP2
SCHEMBL16213220 0.85 EED (0.64) EEDRBBP4SUZ12EZH2AEBP2
SCHEMBL16212973 0.85 EZH2 (0.65) EEDRBBP4SUZ12EZH2AEBP2
SCHEMBL17713651 0.84 EED (0.56) EEDRBBP4SUZ12EZH2AEBP2
SCHEMBL17713654 0.84 EED (0.51) EEDRBBP4SUZ12EZH2AEBP2
SCHEMBL17713628 0.84 EZH2 (0.68) EEDRBBP4SUZ12EZH2AEBP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3212639-A1 ENHANCER OF ZESTE HOMOLOG 2 INHIBITORS Glaxosmithkline Intellectual Property (No. 2) Limited (GB) 2017-09-06 EP claimed
WO-2016066697-A1 ENHANCER OF ZESTE HOMOLOG 2 INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED (GB) 2016-05-06 WO claimed
EP-3212639-A1 ENHANCER OF ZESTE HOMOLOG 2 INHIBITORS Glaxosmithkline Intellectual Property (No. 2) Limited (GB) 2017-09-06 EP disclosed
WO-2016066697-A1 ENHANCER OF ZESTE HOMOLOG 2 INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED (GB) 2016-05-06 WO disclosed