SCHEMBL177310

SCHEMBL177310

CCOC(=O)c1cccc(N)c1O

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.72
HSD17B10 Q99714 4/20 0.72
TSHR P16473 1/20 0.61
CDC25B P30305 4/20 0.56
MMP2 P08253 1/20 0.55
CA12 O43570 3/20 0.53
CA1 P00915 3/20 0.53
CA2 P00918 3/20 0.53
CA7 P43166 3/20 0.53
CA9 Q16790 3/20 0.53
CA14 Q9ULX7 3/20 0.53
GAA P10253 3/20 0.49
MAPT P10636 2/20 0.49
HPGD P15428 2/20 0.49
ALOX15 P16050 1/20 0.49
RAB9A P51151 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
KDM4E B2RXH2 1/20 0.49
POLB P06746 1/20 0.49
CYP1A2 P05177 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10571657 0.87 TSHR (0.73) ALDH1A1HSD17B10TSHRCDC25BCA12
SCHEMBL2927900 0.87 ALDH1A1 (0.64) ALDH1A1HSD17B10TSHRCDC25BMMP2
SCHEMBL28994824 0.84 ALDH1A1 (0.56) ALDH1A1HSD17B10TSHRCDC25BMMP2
SCHEMBL2925689 0.84 ALDH1A1 (0.74) ALDH1A1HSD17B10TSHRCDC25BCA12
SCHEMBL717606 0.84 ALDH1A1 (0.74) ALDH1A1HSD17B10TSHRCDC25BCA12
SCHEMBL27883893 0.84 ALDH1A1 (0.59) ALDH1A1HSD17B10TSHRCDC25BCA12
Ethyl Anthranilate SCHEMBL30055126 0.84 ALDH1A1 (1.00) ALDH1A1HSD17B10TSHRCDC25BGAA
Ethyl Anthranilate SCHEMBL34474 0.84 ALDH1A1 (1.00) ALDH1A1HSD17B10TSHRCDC25BGAA
SCHEMBL2894636 0.83 ALDH1A1 (0.72) ALDH1A1HSD17B10TSHRCDC25BCA12
Ethyl Anthranilate SCHEMBL1396081 0.82 ALDH1A1 (0.96) ALDH1A1HSD17B10TSHRCDC25BGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 93 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003016615-A1 SINGLE BATH PROCESS FOR BLEACHING AND DYEING TEXTILES NOVOZYMES NORTH AMERICA, INC. (US) 2003-02-27 WO claimed
EP-2708223-B1 DYEING AGENT AND USE FOR SAME AMANO ENZYME INC (JP) 2017-02-01 EP disclosed
CN-103980309-B Casr agonist AJINOMOTO K. K. (JP) 2016-04-06 CN disclosed
EP-2345636-B1 CASR AGONIST AJINOMOTO KK (JP) 2016-03-30 EP disclosed
EP-2627652-B1 PYRIDYL BENZOXAZINE DERIVATIVES, PHARMACEUTICAL COMPOSITION COMPRISING THE SAME, AND USE THEREOF DAE WOONG PHARMA (KR) 2015-12-16 EP disclosed
EP-2627652-B1 PYRIDYL BENZOXAZINE DERIVATIVES, PHARMACEUTICAL COMPOSITION COMPRISING THE SAME, AND USE THEREOF DAE WOONG PHARMA (KR) 2015-12-16 EP disclosed
US-9174932-B2 CaSR agonists AJINOMOTO CO., INC. (JP) 2015-11-03 US disclosed
CN-103153990-B Novel pyridyl benzoxazine derivatives, pharmaceutical composition comprising the same, and use thereof DAE WOONG PHARMA 2015-06-17 CN disclosed
CN-101983197-B A novel benzoxazine benzimidazole derivative, a pharmaceutical composition comprising the same, and a use thereof DAE WOONG PHARMA 2015-04-22 CN disclosed
EP-2264031-B1 A NOVEL BENZOXAZINE BENZIMIDAZOLE DERIVATIVE, A PHARMACEUTICAL COMPOSITION COMPRISING THE SAME, AND A USE THEREOF DAE WOONG PHARMA (KR) 2015-04-15 EP disclosed
US-6207693-B1 Benzamide derivatives having a vasopressin antagonistic activity FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-03-27 US disclosed
US-6036729-A DYEING, SOAKING MATERIAL WITH NAPHTHOLS, HYDROGEN PEROXIDE AND ENZYMES OF PEROXIDASE OR OXIDASE NOVO NORDISK A/S (DK) 2000-03-14 US disclosed
US-5972042-A DYEING SYSTEM WHICH COMPRISES ONE OR MORE MONO-, DI- OR POLYCYCLIC AROMATIC OR HETEROAROMATIC COMPOUNDS, AND HYDROGEN PEROXIDE SOURCE AND ENZYME EXHIBITING PEROXIDASE ACTIVITY OR ENZYME EXHIBITING OXIDASE ACTIVITY NOVO NORDISK A/S (DE) 1999-10-26 US disclosed
EP-0946519-A1 BENZAMIDE DERIVATIVES HAVING A VASOPRESSIN ANTAGONISTIC ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-10-06 EP disclosed
US-5925148-A TREATING IN AQUEOUS DYE LIQUOR WITH SYSTEM COMPRISING SUBSTITUTED AROMATIC COMPOUND, HYDROGEN PEROXIDE SOURCE AND PEROXIDASE ENZYME AND/OR OXIDASE ENZYME NOVO NORDISK A/S (DK) 1999-07-20 US disclosed
EP-0870082-A1 ENZYMATIC METHOD FOR DYEING NOVO NORDISK BIOCHEM NORTH AMERICA (US) 1998-10-14 EP disclosed
WO-1998024771-A1 BENZAMIDE DERIVATIVES HAVING A VASOPRESSIN ANTAGONISTIC ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-06-11 WO disclosed
WO-1997023684-A1 ENZYMATIC METHOD FOR DYEING NOVO NORDISK BIOCHEM NORTH AMERICA, INC. (US) 1997-07-03 WO disclosed
US-4461827-A Color photographic recording material containing a non-diffusible dye releaser from which a complexible azo dye is released during development AGFA-GEVAERT AKTIENGESELLSCHAFT (DE) 1984-07-24 US disclosed
US-4036951-A SUNSCREEN AGENTS SYNERGISTICS, INC. (US) 1977-07-19 US disclosed