SCHEMBL17733741

SCHEMBL17733741

Nc1cc(Cl)nc(NC[C@H]2CC[C@@H](N)CC2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.49
PAK4 O96013 2/20 0.42
PAK1 Q13153 2/20 0.42
VCP P55072 6/20 0.37
CCNK O75909 1/20 0.36
CDK9 P50750 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MAPK1 P28482 1/20 0.36
PTGER4 P35408 1/20 0.35
FLT3 P36888 2/20 0.35
TYRO3 Q06418 2/20 0.35
MERTK Q12866 2/20 0.35
GAS6 Q14393 2/20 0.35
AXL P30530 1/20 0.35
CCNB2 O95067 1/20 0.34
CCNE2 O96020 1/20 0.34
CDK1 P06493 1/20 0.34
CDK4 P11802 1/20 0.34
CCNB1 P14635 1/20 0.34
CCND1 P24385 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9885082 1.00 HRH4 (0.49) HRH4PAK4PAK1VCPCCNK
SCHEMBL9885067 0.88 HRH4 (0.49) HRH4VCPKDM4EMAPK1CDK1
SCHEMBL16790179 0.88 HRH4 (0.49) HRH4VCPKDM4EMAPK1CDK1
SCHEMBL13668600 0.88 HRH4 (0.49) HRH4VCPKDM4EMAPK1CDK1
SCHEMBL9884988 0.84 HRH4 (0.45) HRH4PAK4PAK1CDK9CCNT1
SCHEMBL13667224 0.82 VCP (0.57) VCP
SCHEMBL17639929 0.81 HRH4 (0.44) HRH4VCPCDK9CDK2CCNT1
SCHEMBL17639934 0.81 HRH4 (0.44) HRH4VCPCDK9CDK2CCNT1
SCHEMBL13683502 0.79 HRH4 (0.46) HRH4VCPCCNKCDK9KDM4E
SCHEMBL9885050 0.79 HRH4 (0.46) HRH4VCPCCNKCDK9KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1890703-B1 PYRIMIDINE COMPOUNDS AS CHEMOKINE RECEPTORS INHIBITORS TAIGEN BIOTECHNOLOGY CO LTD (TW) 2016-05-11 EP disclosed