SCHEMBL17734089

SCHEMBL17734089

C1=CCNC(N2CCOCC2)=C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
LMNA P02545 2/20 0.35
KMT2A Q03164 3/20 0.35
HTT P42858 3/20 0.34
GAA P10253 1/20 0.33
MEN1 O00255 2/20 0.32
MAPT P10636 2/20 0.32
NPC1 O15118 1/20 0.32
CYP1A2 P05177 1/20 0.32
RAB9A P51151 1/20 0.32
PIK3CA P42336 4/20 0.32
POLB P06746 2/20 0.32
KDM4E B2RXH2 2/20 0.32
TP53 P04637 2/20 0.32
USP2 O75604 1/20 0.32
ALOX15 P16050 1/20 0.32
MAPK1 P28482 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PIK3R1 P27986 2/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17067817 0.78 KDM4E (0.42) ALDH1A1KDM4EUSP2
SCHEMBL30724578 0.69 LMNA (0.35) ALDH1A1LMNAKMT2AHTTGAA
SCHEMBL17787710 0.68 LMNA (0.34) ALDH1A1LMNAKMT2AHTTGAA
SCHEMBL17655487 0.67 MAPT (0.38) ALDH1A1LMNAKMT2AHTTMEN1
SCHEMBL15647482 0.64 LMNA (0.34) ALDH1A1LMNAKMT2AHTTGAA
SCHEMBL883891 0.64 LMNA (0.34) ALDH1A1LMNAKMT2AHTTGAA
SCHEMBL30425332 0.63 LMNA (0.36) ALDH1A1LMNAKMT2AHTTGAA
SCHEMBL19027031 0.62 MAPT (0.35) LMNAKMT2AHTTGAAMEN1
SCHEMBL19027124 0.62 GAA (0.40) ALDH1A1KMT2AGAAMEN1MAPT
SCHEMBL229286 0.60 LMNA (0.57) ALDH1A1LMNAKMT2AHTTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611777-B1 N-(4-{[PYRIDIN-3-YL-METHYL)CARBAMOYL]AMINO}BENZENE-SULFONE DERIVATIVES AS NAMPT INHIBITORS FOR THERAPY OF DISEASES SUCH AS CANCER FORMA TM LLC (US) 2016-05-11 EP disclosed