SCHEMBL17745705

SCHEMBL17745705

COc1cc2nccc(Oc3ccc(NC(=O)Oc4nn(C)c(=O)[nH]c4=O)cc3F)c2cc1OC

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 14/20 0.77
AXL P30530 12/20 0.77
PDGFRA P16234 1/20 0.55
KDR P35968 2/20 0.55
AURKA O14965 1/20 0.54
JAK2 O60674 1/20 0.54
RPS6KA5 O75582 1/20 0.54
ABL1 P00519 1/20 0.54
INSR P06213 1/20 0.54
LCK P06239 1/20 0.54
RET P07949 1/20 0.54
IGF1R P08069 1/20 0.54
KIT P10721 1/20 0.54
PIM1 P11309 1/20 0.54
FGFR1 P11362 1/20 0.54
SRC P12931 1/20 0.54
PRKACA P17612 1/20 0.54
RPS6KB1 P23443 1/20 0.54
JAK1 P23458 1/20 0.54
MAPK3 P27361 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16089972 0.87 MET (1.00) METAXL
SCHEMBL17745593 0.84 MET (0.78) METAXL
SCHEMBL17745532 0.84 MET (0.78) METAXL
SCHEMBL17745536 0.83 MET (0.68) METAXL
SCHEMBL17745650 0.82 MET (0.78) METAXL
SCHEMBL17745622 0.82 MET (0.57) METAXL
SCHEMBL17745621 0.82 AXL (0.79) METAXLPDGFRAKDR
SCHEMBL17745550 0.82 MET (0.79) METAXL
SCHEMBL17745645 0.82 AXL (0.79) METAXL
SCHEMBL17745537 0.82 MET (0.79) METAXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2780338-B1 URACIL DERIVATIVES AS AXL AND C-MET KINASE INHIBITORS IGNYTA INC (US) 2016-11-09 EP claimed