SCHEMBL1775181

SCHEMBL1775181

NS(=O)(=O)c1cccc(C[O])c1

nearest known ligand 0.64

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA2 P00918 12/20 0.64
CA1 P00915 9/20 0.64
CA9 Q16790 8/20 0.55
CA12 O43570 7/20 0.55
CA14 Q9ULX7 4/20 0.55
CA4 P22748 3/20 0.55
CA5A P35218 3/20 0.48
CA7 P43166 3/20 0.48
CA6 P23280 2/20 0.48
CA5B Q9Y2D0 2/20 0.48
CA3 P07451 1/20 0.48
PLA2G7 Q13093 1/20 0.48
CA13 Q8N1Q1 1/20 0.48
MAPT P10636 1/20 0.45
HTR6 P50406 1/20 0.44
NOS1 P29475 1/20 0.44
ALDH1A1 P00352 1/20 0.44
PKM P14618 1/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1795003 0.83 CA2 (0.64) CA2CA1CA9CA12CA14
SCHEMBL246236 0.82 CA2 (0.61) CA2CA1CA9CA12CA14
SCHEMBL2181186 0.82 CA2 (0.61) CA2CA1CA9CA12CA14
SCHEMBL2005567 0.82 CA2 (0.61) CA2CA1CA9CA12CA14
SCHEMBL3446128 0.82 CA2 (0.61) CA2CA1CA9CA12CA14
Hydrochloric Acid SCHEMBL19272459 0.82 CA2 (0.64) CA2CA1CA9CA12CA14
SCHEMBL185757 0.82 CA2 (0.61) CA2CA1CA9CA12CA14
SCHEMBL7179836 0.82 CA2 (0.61) CA2CA1CA9CA12CA14
SCHEMBL16410190 0.82 CA2 (0.61) CA2CA1CA9CA12CA14
SCHEMBL28223875 0.82 CA2 (0.61) CA2CA1CA9CA12CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7943637-B2 Thienopyridine derivatives and the use thereof as HSP90 modulators MERCK PATENT GMBH (DE) 2011-05-17 US disclosed
US-20090054452-A1 Thienopyridine Derivatives and the Use Thereof as Hsp90 Modulators MERCK PATENT GMBH (DE) 2009-02-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090054452-A1 Thienopyridine Derivatives and the Use Thereof as Hsp90 Modulators HSP90AA1, HSP90AB1, HSP90AB2P CA2 3625/4885CA1 4690/4885CA9 4875/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.