SCHEMBL17772010

SCHEMBL17772010

Cc1ccccc1N1CCN(C(=O)CNc2c(-c3ccc(N4CCCC4)cc3)nc3cnccn23)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 13/20 0.53
MAPT P10636 8/20 0.53
KDM4E B2RXH2 7/20 0.53
NPC1 O15118 2/20 0.53
RAB9A P51151 2/20 0.53
RXFP1 Q9HBX9 2/20 0.51
ALDH1A1 P00352 4/20 0.48
CASP1 P29466 3/20 0.48
CASP7 P55210 3/20 0.48
HSD17B10 Q99714 3/20 0.48
HPGD P15428 2/20 0.48
ALOX15 P16050 1/20 0.48
TP53 P04637 4/20 0.47
ALOX5 P09917 1/20 0.46
BRD4 O60885 3/20 0.45
TDP1 Q9NUW8 2/20 0.42
CDK9 P50750 1/20 0.42
HTR1A P08908 1/20 0.40
HTR1D P28221 1/20 0.40
HTR1B P28222 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10048672 0.94 GAA (0.52) GAAMAPTKDM4ENPC1RAB9A
SCHEMBL14963805 0.91 GAA (0.49) GAAMAPTKDM4ENPC1RAB9A
SCHEMBL10120181 0.91 GAA (0.49) GAAMAPTKDM4ENPC1RAB9A
SCHEMBL10120322 0.91 GAA (0.46) GAAMAPTKDM4ENPC1RAB9A
SCHEMBL14963802 0.90 GAA (0.48) GAAMAPTKDM4ENPC1RAB9A
SCHEMBL10120308 0.90 GAA (0.47) GAAMAPTKDM4ENPC1RAB9A
SCHEMBL10120622 0.90 GAA (0.50) GAAMAPTKDM4ENPC1RAB9A
SCHEMBL15179400 0.90 KDM4E (0.48) GAAMAPTKDM4ENPC1RAB9A
SCHEMBL15179447 0.89 KDM4E (0.53) GAAMAPTKDM4ENPC1RAB9A
SCHEMBL15179449 0.89 GAA (0.46) GAAMAPTKDM4ENPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2601194-B1 FUSED-IMIDAZOYL COMPOUNDS USEFUL AS ANTIMICROBIAL AGENTS MERCK SHARP & DOHME (US) 2016-05-25 EP disclosed