SCHEMBL10120181

SCHEMBL10120181

Cc1ccc(C)c(N2CCN(C(=O)CNc3c(-c4ccc(N5CCCC5)cc4)nc4cnccn34)CC2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 11/20 0.49
MAPT P10636 9/20 0.49
KDM4E B2RXH2 8/20 0.49
ALDH1A1 P00352 5/20 0.47
CASP1 P29466 3/20 0.47
CASP7 P55210 3/20 0.47
HPGD P15428 2/20 0.47
HSD17B10 Q99714 2/20 0.47
ALOX15 P16050 1/20 0.47
RXFP1 Q9HBX9 1/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
TP53 P04637 3/20 0.46
ALOX5 P09917 1/20 0.45
BRD4 O60885 2/20 0.43
MEN1 O00255 1/20 0.43
TSHR P16473 1/20 0.43
KMT2A Q03164 1/20 0.43
LMNA P02545 2/20 0.42
TDP1 Q9NUW8 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15179447 0.92 KDM4E (0.53) GAAMAPTKDM4EALDH1A1CASP1
SCHEMBL17772010 0.91 GAA (0.53) GAAMAPTKDM4EALDH1A1CASP1
SCHEMBL10048672 0.88 GAA (0.52) GAAMAPTKDM4EALDH1A1CASP1
SCHEMBL10049161 0.87 GAA (0.52) GAAMAPTKDM4EALDH1A1CASP1
SCHEMBL10049160 0.86 GAA (0.52) GAAMAPTKDM4EALDH1A1CASP1
SCHEMBL10049172 0.86 GAA (0.52) GAAMAPTKDM4EALDH1A1CASP1
SCHEMBL10120323 0.85 GAA (0.49) GAAMAPTKDM4EALDH1A1CASP1
SCHEMBL10048728 0.85 NCF1 (0.46) GAAMAPTKDM4EALDH1A1CASP1
SCHEMBL14963805 0.85 GAA (0.49) GAAMAPTKDM4EALDH1A1CASP1
SCHEMBL10120322 0.84 GAA (0.46) GAAMAPTKDM4EALDH1A1CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012018662-A2 FUSED-IMIDAZOYL COMPOUNDS USEFUL AS ANTIMICROBIAL AGENTS SCHERING CORPORATION (US) 2012-02-09 WO disclosed