SCHEMBL17797397

SCHEMBL17797397

CCCOc1ccc(-c2nc(-c3ccc4oc(C5(NC(=O)OC(C)(C)C)COC(C)(C)OC5)cc4c3)no2)cc1OC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 10/20 0.45
S1PR3 Q99500 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
MAPT P10636 4/20 0.39
TPH1 P17752 2/20 0.38
KDM4E B2RXH2 2/20 0.36
HSD17B10 Q99714 2/20 0.36
MEN1 O00255 1/20 0.36
TP53 P04637 1/20 0.36
TSHR P16473 1/20 0.36
XBP1 P17861 1/20 0.36
PPARG P37231 1/20 0.36
KMT2A Q03164 1/20 0.36
NCOA2 Q15596 1/20 0.36
LMNA P02545 2/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17797399 0.93 S1PR1 (0.45) S1PR1S1PR3MAPTKDM4EHSD17B10
SCHEMBL15662510 0.93 MAPT (0.45) S1PR1S1PR3SMN1; SMN2MAPTTPH1
SCHEMBL177105 0.92 S1PR1 (0.55) S1PR1S1PR3
SCHEMBL15662798 0.92 SMN1; SMN2 (0.49) S1PR1S1PR3SMN1; SMN2MAPTTPH1
SCHEMBL17797432 0.91 S1PR1 (0.52) S1PR1S1PR3SMN1; SMN2MAPTKDM4E
SCHEMBL178195 0.91 S1PR1 (0.46) S1PR1S1PR3SMN1; SMN2MAPTTPH1
SCHEMBL17797433 0.90 S1PR1 (0.44) S1PR1S1PR3
SCHEMBL17797420 0.90 S1PR1 (0.42) S1PR1S1PR3MAPTTP53
SCHEMBL15662730 0.89 TPH1 (0.40) S1PR1S1PR3SMN1; SMN2MAPTTPH1
SCHEMBL15662834 0.85 SMN1; SMN2 (0.52) S1PR1S1PR3SMN1; SMN2MAPTTPH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2344484-B1 S1P RECEPTORS MODULATORS AND USE THEREOF AKAAL PHARMA PTY LTD (AU) 2016-06-08 EP disclosed