SCHEMBL17801360

SCHEMBL17801360

Clc1cc2sc(-c3cccnc3)nc2cn1.[Ar]

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.58
RAB9A P51151 1/20 0.58
CYP19A1 P11511 3/20 0.47
CYP2A6 P11509 6/20 0.46
PIK3CD O00329 1/20 0.44
PIP5K1C O60331 1/20 0.44
PIK3CA P42336 1/20 0.44
PI4KA P42356 1/20 0.44
PI4KB Q9UBF8 1/20 0.44
ALOX5 P09917 1/20 0.43
KDM4E B2RXH2 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.40
AXL P30530 1/20 0.40
PBRM1 Q86U86 1/20 0.40
MKNK1 Q9BUB5 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40
CLK1 P49759 1/20 0.39
DYRK1A Q13627 1/20 0.39
ILK Q13418 1/20 0.39
CYP3A4 P08684 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17801257 0.99 NPC1 (0.60) NPC1RAB9ACYP19A1CYP2A6PIK3CD
SCHEMBL17801340 0.83 NPC1 (0.61) NPC1RAB9ACYP19A1CYP2A6PIK3CD
SCHEMBL17801198 0.82 RAB9A (0.60) NPC1RAB9ACYP19A1CYP2A6PIK3CD
SCHEMBL17801374 0.78 NPC1 (0.56) NPC1RAB9ACYP19A1CYP2A6PIK3CD
SCHEMBL17801186 0.77 RAB9A (0.62) NPC1RAB9ACYP19A1CYP2A6PIK3CD
SCHEMBL17801309 0.77 NPC1 (0.55) NPC1RAB9APIK3CDPIP5K1CPIK3CA
SCHEMBL20519963 0.77 RAB9A (0.76) NPC1RAB9ACYP19A1CYP2A6PIK3CD
SCHEMBL24366502 0.77 NPC1 (0.66) NPC1RAB9ACYP19A1CYP2A6ALOX5
SCHEMBL21589907 0.76 APP (0.43) NPC1RAB9A
SCHEMBL17812983 0.76 NPC1 (0.59) NPC1RAB9ACYP19A1PIK3CDPIP5K1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3227301-A1 BICYCLIC COMPOUNDS AS PEST CONTROL AGENTS Bayer CropScience AG (DE) 2017-10-11 EP disclosed
WO-2016087417-A1 BICYCLIC COMPOUNDS AS PEST CONTROL AGENTS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2016-06-09 WO disclosed