SCHEMBL17801378

SCHEMBL17801378

CC(C)(C)N(C(=O)O)c1cc2sc(-c3cccnc3)nc2cn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
CYP3A4 P08684 3/20 0.41
CYP1A2 P05177 2/20 0.41
LMNA P02545 2/20 0.41
CYP2C19 P33261 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
PIK3CA P42336 1/20 0.40
PIK3CG P48736 1/20 0.40
KDM4E B2RXH2 7/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ALOX5 P09917 1/20 0.39
ALDH1A1 P00352 3/20 0.39
GFER P55789 1/20 0.39
CDC7 O00311 1/20 0.38
DBF4 Q9UBU7 1/20 0.38
MAPT P10636 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17803434 0.81 CYP3A4 (0.43) NPC1RAB9ACYP3A4CYP1A2LMNA
SCHEMBL17801309 0.77 NPC1 (0.55) NPC1RAB9ACYP3A4CYP1A2LMNA
SCHEMBL17801310 0.74 NPC1 (0.51) NPC1RAB9ACYP3A4CYP1A2LMNA
SCHEMBL20519387 0.74 NPC1 (0.51) NPC1RAB9ACYP3A4CYP1A2LMNA
SCHEMBL16652413 0.74 CYP3A4 (0.45) NPC1RAB9ACYP3A4CYP1A2LMNA
SCHEMBL17801346 0.74 NPC1 (0.41) NPC1RAB9ACYP3A4CYP1A2LMNA
SCHEMBL17801295 0.73 DYRK1A (0.54) NPC1RAB9ACYP3A4CYP1A2LMNA
SCHEMBL17816547 0.73 RAB9A (0.44) NPC1RAB9ACYP3A4CYP1A2LMNA
SCHEMBL17801340 0.72 NPC1 (0.61) NPC1RAB9ACYP3A4CYP1A2LMNA
SCHEMBL17801688 0.72 KDM4E (0.74) NPC1RAB9ACYP3A4CYP1A2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3227301-A1 BICYCLIC COMPOUNDS AS PEST CONTROL AGENTS Bayer CropScience AG (DE) 2017-10-11 EP disclosed
WO-2016087417-A1 BICYCLIC COMPOUNDS AS PEST CONTROL AGENTS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2016-06-09 WO disclosed