SCHEMBL17803166

SCHEMBL17803166

O=C(O)/C(Cl)=N\Nc1ccc(C(F)(F)F)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.49
RAB9A P51151 2/20 0.46
NPC1 O15118 1/20 0.46
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
PKM P14618 1/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
KMT2A Q03164 1/20 0.44
RELA Q04206 1/20 0.44
ATM Q13315 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KIF11 P52732 1/20 0.42
PTPN1 P18031 1/20 0.42
TGM2 P21980 1/20 0.42
KCNQ3 O43525 1/20 0.42
KCNQ2 O43526 1/20 0.42
KCNE1 P15382 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17803167 1.00 EPHX2 (0.49) EPHX2RAB9ANPC1MEN1ALDH1A1
SCHEMBL11765759 0.81 CA1 (0.55) RAB9ANPC1MEN1ALDH1A1GAA
SCHEMBL11765765 0.81 CA1 (0.55) RAB9ANPC1MEN1ALDH1A1GAA
SCHEMBL5843519 0.80 EPHX2 (0.49) EPHX2RAB9ANPC1MEN1ALDH1A1
SCHEMBL2383847 0.80 KMT2A (0.56) EPHX2RAB9ANPC1MEN1ALDH1A1
SCHEMBL2383845 0.80 KMT2A (0.56) EPHX2RAB9ANPC1MEN1ALDH1A1
SCHEMBL9102812 0.80 KMT2A (0.56) EPHX2RAB9ANPC1MEN1ALDH1A1
SCHEMBL9723601 0.79 CA1 (0.62) EPHX2MEN1GAAMAPTKMT2A
SCHEMBL9723609 0.79 CA1 (0.62) EPHX2MEN1GAAMAPTKMT2A
SCHEMBL17803163 0.79 NPSR1 (0.58) RAB9ANPC1MEN1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3227282-A1 NOVEL PIPERIDINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2017-10-11 EP disclosed
WO-2016087352-A1 NOVEL PIPERIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2016-06-09 WO disclosed