SCHEMBL17825837

SCHEMBL17825837

NC(=O)C(c1ccccc1)n1ccnn1

nearest known ligand 0.59

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 19/20 0.59
CYP1A1 P04798 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11499232 0.80 TSHR (0.41) CYP19A1
SCHEMBL4592845 0.79 SMN1; SMN2 (0.44) CYP19A1
SCHEMBL5865736 0.74 CYP19A1 (1.00) CYP19A1CYP1A1
SCHEMBL9756477 0.74 CYP19A1 (0.56) CYP19A1CYP1A1
SCHEMBL5782527 0.73 SMN1; SMN2 (0.45)
SCHEMBL27494651 0.72 CYP19A1 (0.57) CYP19A1
SCHEMBL5972481 0.72 CYP19A1 (0.57) CYP19A1
SCHEMBL3579264 0.72 CYP19A1 (0.53) CYP19A1CYP1A1
SCHEMBL11015925 0.72 CYP19A1 (0.67) CYP19A1CYP1A1
SCHEMBL29471930 0.72 CYP19A1 (0.67) CYP19A1CYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3229801-A1 FACTOR IXA INHIBITORS Merck Sharp & Dohme Corp. (US) 2017-10-18 EP disclosed
WO-2016094260-A1 FACTOR IXA INHIBITORS MERCK SHARP & DOHME CORP. (US) 2016-06-16 WO disclosed
CN-101223143-A 3-cyanoquinoline inhibitors of TPL2 kinase and methods of making and using the same WYETH CORP (US) 2008-07-16 CN disclosed