SCHEMBL17826183

SCHEMBL17826183

C=C(c1ccc(-c2cncc(-c3nnc(-c4ccccc4OCCN)o3)n2)cc1)N(C)C

nearest known ligand 0.62

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
ATR Q13535 20/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17826177 0.93 ATR (0.53) ATR
SCHEMBL17826208 0.91 ATR (0.51) ATR
SCHEMBL17826206 0.90 ATR (0.49) ATR
SCHEMBL16420734 0.89 ATR (0.78) ATR
SCHEMBL17826191 0.87 ATR (0.45) ATR
SCHEMBL17826143 0.84 ATR (0.43) ATR
SCHEMBL17826170 0.83 ATR (0.48) ATR
SCHEMBL17826163 0.83 ATR (0.57) ATR
SCHEMBL17826139 0.83 ATR (0.45) ATR
SCHEMBL17826111 0.83 NPC1 (0.48) ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9365557-B2 Substituted pyrazin-2-amines as inhibitors of ATR kinase VERTEX PHARMACEUTICALS INCORPORATED (US) 2016-06-14 US disclosed