SCHEMBL17832244

SCHEMBL17832244

O=Cc1ccc(N2CCC(c3ccc(OC(F)(F)F)cc3)CC2)nc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCAT P04180 2/20 0.44
DGAT1 O75907 1/20 0.42
GRM2 Q14416 1/20 0.42
CHRM4 P08173 2/20 0.41
CACNA1G O43497 1/20 0.40
CACNA1H O95180 1/20 0.40
CACNA1I Q9P0X4 1/20 0.40
EPHX2 P34913 1/20 0.40
BCHE P06276 1/20 0.40
ACHE P22303 1/20 0.40
BACE1 P56817 1/20 0.40
SCN9A Q15858 1/20 0.40
FAAH O00519 1/20 0.39
EGLN1 Q9GZT9 1/20 0.38
BRD4 O60885 4/20 0.38
SMO Q99835 1/20 0.38
AR P10275 1/20 0.38
KCNH2 Q12809 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ABL1 P00519 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17832235 0.86 FAAH (0.47) DGAT1CHRM4EPHX2FAAHKCNH2
SCHEMBL17832257 0.86 SCN9A (0.44) LCATGRM2EPHX2SCN9AFAAH
SCHEMBL17832319 0.83 BCHE (0.44) CACNA1GCACNA1HCACNA1IBCHEACHE
SCHEMBL17832250 0.82 ACACB (0.51)
SCHEMBL31732104 0.82 FAAH (0.47) LCATGRM2CHRM4EPHX2SCN9A
SCHEMBL17832239 0.80 ACACB (0.39) CHRM4EPHX2FAAHKCNH2
SCHEMBL21620073 0.78 KDM4E (0.46) DGAT1SMOKDM4EABL1LMNA
SCHEMBL17832273 0.78 CACNA1B (0.40) CACNA1GCACNA1HCACNA1IEPHX2BCHE
SCHEMBL17832304 0.78 CHRM4 (0.42) LCATCHRM4CACNA1GCACNA1HCACNA1I
SCHEMBL14893604 0.77 BCHE (0.56) GRM2BCHEACHEBACE1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170334927-A1 Nitroimidazole Compound, Preparation Method Therefor And Use Thereof In Drug Manufacturing SHANGHAI SUN-SAIL PHARMACEUTICAL SCIENCE & TECHNOLOGY CO., LTD. (CN) 2017-11-23 US disclosed
US-20170334927-A1 Nitroimidazole Compound, Preparation Method Therefor And Use Thereof In Drug Manufacturing SHANGHAI SUN-SAIL PHARMACEUTICAL SCIENCE & TECHNOLOGY CO., LTD. (CN) 2017-11-23 US disclosed
WO-2016091207-A1 NITROMIDAZOLE COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF IN DRUG MANUFACTURING 上海阳帆医药科技有限公司 2016-06-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170334927-A1 Nitroimidazole Compound, Preparation Method Therefor And Use Thereof In Drug Manufacturing NISCH, CYP51A1, CYP4F11 LCAT 3270/4885DGAT1 2403/4885GRM2 4732/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.