SCHEMBL17845772

SCHEMBL17845772

CCNC(C)c1ncc(Br)cn1

nearest known ligand 0.38

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
GBA1 P04062 1/20 0.32
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24774903 0.81 NPC1 (0.39) NPC1RAB9AGBA1
SCHEMBL31064460 0.72 IDH1 (0.38)
SCHEMBL11089872 0.71 NPC1 (0.41) NPC1RAB9AGBA1KDM4E
SCHEMBL20714561 0.71 NPC1 (0.47) NPC1RAB9A
SCHEMBL23507732 0.71 NPC1 (0.47) NPC1RAB9A
SCHEMBL17845775 0.69
SCHEMBL20303574 0.69 ALDH1A1 (0.36) NPC1RAB9AKDM4E
SCHEMBL27875523 0.69 KDM4E (0.37) NPC1RAB9AGBA1KDM4E
SCHEMBL13981511 0.68 KDM4E (0.39) NPC1RAB9AKDM4E
SCHEMBL29251485 0.68 MAPK10 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016095205-A1 HETEROARYL OREXIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-06-23 WO disclosed