SCHEMBL17845779

SCHEMBL17845779

[CH2]Cc1ccc(C#N)cn1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.42
ALDH1A1 P00352 5/20 0.42
L3MBTL1 Q9Y468 3/20 0.42
MBOAT4 Q96T53 1/20 0.39
LMNA P02545 1/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 3/20 0.36
HTT P42858 2/20 0.36
CYP19A1 P11511 1/20 0.36
EGLN2 Q96KS0 1/20 0.36
CYP2A6 P11509 1/20 0.34
LOXL2 Q9Y4K0 1/20 0.34
XDH P47989 1/20 0.34
GRM5 P41594 1/20 0.34
FFAR1 O14842 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1042523 0.84 KDM4E (0.40) KDM4EALDH1A1L3MBTL1MBOAT4LMNA
SCHEMBL453493 0.83 KDM4E (0.42) KDM4EALDH1A1L3MBTL1MBOAT4LMNA
SCHEMBL2633134 0.83 CYP2A6 (0.48) KDM4EALDH1A1L3MBTL1MBOAT4LMNA
SCHEMBL507552 0.79 KDM4E (0.42) KDM4EALDH1A1L3MBTL1MBOAT4LMNA
SCHEMBL17266360 0.79 KDM4E (0.42) KDM4EALDH1A1L3MBTL1MBOAT4LMNA
SCHEMBL23171396 0.79 MEN1 (0.43) KDM4EALDH1A1L3MBTL1MBOAT4LMNA
SCHEMBL4851284 0.79 LOXL2 (0.48) KDM4EALDH1A1L3MBTL1MBOAT4LMNA
SCHEMBL450943 0.79 KDM4E (0.42) KDM4EALDH1A1L3MBTL1MBOAT4LMNA
SCHEMBL6245066 0.79 KDM4E (0.42) KDM4EALDH1A1L3MBTL1MBOAT4LMNA
SCHEMBL450944 0.79 NOTUM (0.45) KDM4EALDH1A1L3MBTL1MBOAT4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016095205-A1 HETEROARYL OREXIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-06-23 WO disclosed