SCHEMBL17848660

SCHEMBL17848660

CC1(Oc2ccc(Cl)cc2)CCN(CCOc2ccc3[nH]c(=O)ccc3c2)C1

nearest known ligand 0.63

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 16/20 0.63
KCNH2 Q12809 1/20 0.49
DRD3 P35462 3/20 0.43
DRD4 P21917 1/20 0.42
FLT3 P36888 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17848643 0.94 DRD2 (0.66) DRD2DRD3DRD4
SCHEMBL29944218 0.94 DRD2 (0.66) DRD2DRD3DRD4
SCHEMBL17848387 0.85 DRD2 (0.79) DRD2DRD3
SCHEMBL17848385 0.82 DRD2 (0.90) DRD2
SCHEMBL17848724 0.80 DRD2 (0.66) DRD2
SCHEMBL17848628 0.80 DRD2 (0.75) DRD2
SCHEMBL17848652 0.80 DRD2 (0.64) DRD2
SCHEMBL17848620 0.79 DRD2 (0.81) DRD2
SCHEMBL17848461 0.78 DRD2 (1.00) DRD2
SCHEMBL17848575 0.78 DRD2 (0.82) DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233077-A1 DOPAMINE D2 RECEPTOR LIGANDS The Broad Institute Inc. (US) 2017-10-25 EP claimed
WO-2016100940-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2016-06-23 WO claimed
EP-3233077-A1 DOPAMINE D2 RECEPTOR LIGANDS The Broad Institute Inc. (US) 2017-10-25 EP disclosed
WO-2016100940-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2016-06-23 WO disclosed