SCHEMBL17850384

SCHEMBL17850384

O=C(Cc1cccc(-n2cc(-c3n[nH]c4ccccc34)nn2)c1)N1CCNCC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 6/20 0.40
ROCK2 O75116 5/20 0.40
IRAK4 Q9NWZ3 3/20 0.40
FLT3 P36888 3/20 0.40
MAP4K4 O95819 2/20 0.40
HIPK2 Q9H2X6 2/20 0.40
CHEK1 O14757 2/20 0.40
MAP2K4 P45985 2/20 0.40
MAPK6 Q16659 2/20 0.40
MAPK8 P45983 2/20 0.40
MAPK9 P45984 2/20 0.40
BMPR1B O00238 1/20 0.40
PLK4 O00444 1/20 0.40
STK25 O00506 1/20 0.40
CIT O14578 1/20 0.40
RIOK3 O14730 1/20 0.40
IKBKB O14920 1/20 0.40
AURKA O14965 1/20 0.40
GAK O14976 1/20 0.40
DCLK1 O15075 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9953146 0.94 POLB (0.42) ROCK1ROCK2IRAK4FLT3MAP4K4
SCHEMBL10194885 0.91 LRRK2 (0.43) FGFR1FLT1MAPK10ITKLRRK2
SCHEMBL10194865 0.91 MAPK10 (0.42) ROCK1ROCK2IRAK4FLT3MAP4K4
SCHEMBL9952065 0.85 CDC7 (0.46) ROCK1ROCK2IRAK4FLT3MAP4K4
SCHEMBL9952277 0.84 NPC1 (0.44) ROCK2IRAK4FLT3MAP4K4HIPK2
SCHEMBL10194814 0.83 ROCK1 (0.43) ROCK1ROCK2CHEK1MAPK8MAPK10
SCHEMBL9951810 0.82 FKBP1A (0.47) FGFR1FLT1MAPK10ITKLRRK2
SCHEMBL10194847 0.80 MAPT (0.47) ROCK1ROCK2MAPK8FGFR1FLT1
SCHEMBL10194944 0.80 MAPK10 (0.46) ROCK1ROCK2FLT3CHEK1FGFR1
SCHEMBL9952518 0.80 CDC7 (0.44) ROCK1ROCK2IRAK4MAP4K4HIPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655357-B1 INDAZOLYL TRIAZOLE DERIVATIVES AS IRAK INHIBITORS MERCK SERONO SA (CH) 2016-06-22 EP disclosed