SCHEMBL17850437

SCHEMBL17850437

N=C(c1cn(-c2ccc(C3CCNCC3)c(C(F)(F)F)c2)nn1)c1ccccc1N

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ESRRA P11474 12/20 0.47
HTR2C P28335 2/20 0.43
NOTUM Q6P988 3/20 0.39
GPR119 Q8TDV5 1/20 0.38
P2RY14 Q15391 2/20 0.35
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
OPRD1 P41143 1/20 0.35
SIGMAR1 Q99720 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17850412 0.74 ESRRA (0.48) ESRRANOTUMGPR119
SCHEMBL10194980 0.71 HTR2C (0.42) HTR2CNOTUMP2RY14ADRA2AADRA2B
SCHEMBL10195750 0.66 ESRRA (0.62) ESRRA
SCHEMBL10196894 0.66 ESRRA (0.56) ESRRA
SCHEMBL10196715 0.66 ESRRA (0.53) ESRRASIGMAR1
SCHEMBL10195780 0.66 ESRRA (0.44) ESRRA
SCHEMBL10194711 0.65 ESRRA (0.60) ESRRA
SCHEMBL14321224 0.65 HTR2C (0.61) HTR2CNOTUM
SCHEMBL27984001 0.65 ESRRA (1.00) ESRRANOTUM
SCHEMBL613612 0.64 HTR2C (1.00) HTR2CSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655357-B1 INDAZOLYL TRIAZOLE DERIVATIVES AS IRAK INHIBITORS MERCK SERONO SA (CH) 2016-06-22 EP disclosed