SCHEMBL17850466

SCHEMBL17850466

Cc1ccc(-c2ccnc(N3CCOCC3)c2)cc1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 10/20 0.55
SMG1 Q96Q15 3/20 0.54
CDK1 P06493 1/20 0.54
CDK2 P24941 1/20 0.54
PIK3CA P42336 2/20 0.52
WNT3A P56704 1/20 0.49
PIK3CD O00329 1/20 0.49
ABL1 P00519 1/20 0.48
CYP2C19 P33261 1/20 0.48
SMO Q99835 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15317749 0.85 ABL1 (0.51) LRRK2SMG1CDK1CDK2PIK3CA
SCHEMBL19998635 0.84 LRRK2 (0.48) LRRK2SMG1CDK1CDK2PIK3CA
SCHEMBL20008239 0.84 BRAF (0.58) LRRK2SMG1CDK1CDK2PIK3CD
SCHEMBL827848 0.83 PIK3CA (0.58) LRRK2SMG1CDK1CDK2PIK3CA
SCHEMBL24512294 0.81 LRRK2 (0.46) LRRK2SMG1CDK1CDK2PIK3CA
SCHEMBL19998588 0.80 USP30 (0.54) LRRK2SMG1CDK1CDK2PIK3CA
SCHEMBL12864090 0.79 CNR2 (0.62) CYP2C19
SCHEMBL16025875 0.79 LRRK2 (0.74) LRRK2
SCHEMBL25666539 0.79 ABL1 (0.74) LRRK2ABL1CYP2C19
SCHEMBL3995999 0.78 LRRK2 (0.52) LRRK2SMG1PIK3CACYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655357-B1 INDAZOLYL TRIAZOLE DERIVATIVES AS IRAK INHIBITORS MERCK SERONO SA (CH) 2016-06-22 EP disclosed