SCHEMBL17866255

SCHEMBL17866255

Cc1cnc(OC(=O)Nc2cnc(OCC(F)(F)F)c(-c3ccc(Cl)cc3)c2)s1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.46
PTGS2 P35354 3/20 0.40
MAPT P10636 4/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
NFKB1 P19838 1/20 0.38
RAB9A P51151 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
KCNH2 Q12809 1/20 0.37
SCN5A Q14524 1/20 0.37
SCN2A Q99250 1/20 0.37
SCN10A Q9Y5Y9 1/20 0.37
CTSA P10619 2/20 0.36
RORA P35398 1/20 0.36
RORC P51449 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2114245 0.86 CNR1 (0.50) CNR1PTGS2MAPTSMN1; SMN2NPSR1
SCHEMBL17866280 0.85 CNR1 (0.46) CNR1PTGS2MAPTSMN1; SMN2NPSR1
SCHEMBL17866274 0.83 CNR1 (0.44) CNR1PTGS2MAPTSMN1; SMN2NPSR1
SCHEMBL17866269 0.83 KCNH2 (0.46) CNR1PTGS2MAPTSMN1; SMN2NPSR1
SCHEMBL17866275 0.83 CNR1 (0.45) CNR1PTGS2MAPTSMN1; SMN2NPSR1
SCHEMBL17866261 0.82 CNR1 (0.47) CNR1PTGS2MAPTSMN1; SMN2NPSR1
SCHEMBL2115870 0.82 CNR1 (0.56) CNR1PTGS2MAPTSMN1; SMN2MEN1
SCHEMBL17866284 0.82 CNR1 (0.48) CNR1PTGS2MAPTSMN1; SMN2NPSR1
SCHEMBL17866271 0.82 CNR1 (0.45) CNR1PTGS2MAPTSMN1; SMN2NPSR1
SCHEMBL17866266 0.82 MAPT (0.45) CNR1PTGS2MAPTSMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2627637-B1 N-PYRIDIN-3-YL OR N-PYRAZIN-2-YL CARBOXAMIDES HOFFMANN LA ROCHE (CH) 2016-06-29 EP claimed