SCHEMBL17874684

SCHEMBL17874684

[2H]c1nc(C)nc([2H])c1-c1cc(NC[C@@H](C)c2cccc3c(C(=O)NC([2H])([2H])[2H])ccnc23)ncn1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 2/20 0.52
FAAH O00519 14/20 0.35
SLC40A1 Q9NP59 1/20 0.33
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
CYP1A2 P05177 2/20 0.32
CYP3A4 P08684 2/20 0.32
HPGD P15428 2/20 0.32
CYP2C19 P33261 2/20 0.32
HSD17B10 Q99714 2/20 0.32
CYP2D6 P10635 1/20 0.32
AURKA O14965 1/20 0.32
RPS6KB1 P23443 1/20 0.32
TSHR P16473 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15328651 0.95 PRKDC (0.53) PRKDCFAAHSLC40A1KDM4EALDH1A1
SCHEMBL16653844 0.95 PRKDC (0.53) PRKDCFAAHSLC40A1KDM4EALDH1A1
SCHEMBL29392854 0.95 PRKDC (0.53) PRKDCFAAHSLC40A1KDM4EALDH1A1
SCHEMBL17634671 0.93 PRKDC (0.60) PRKDCFAAHSLC40A1KDM4EALDH1A1
SCHEMBL17874734 0.91 PRKDC (0.57) PRKDCFAAHSLC40A1KDM4EALDH1A1
SCHEMBL17874765 0.90 PRKDC (0.55) PRKDCFAAHKDM4EALDH1A1CYP1A2
SCHEMBL17874686 0.89 PRKDC (0.54) PRKDCFAAHSLC40A1KDM4EAURKA
SCHEMBL17634601 0.89 PRKDC (0.52) PRKDCFAAHSLC40A1KDM4EALDH1A1
SCHEMBL15328700 0.87 PRKDC (0.63) PRKDCFAAHSLC40A1KDM4EALDH1A1
SCHEMBL16654055 0.87 PRKDC (0.63) PRKDCFAAHSLC40A1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9376448-B2 DNA-PK inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2016-06-28 US disclosed