SCHEMBL17874686

SCHEMBL17874686

[2H]c1nc(C)nc([2H])c1-c1cc(NC[C@@H](C)c2cccc3c(C(N)=O)ccnc23)ncn1

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 2/20 0.54
L3MBTL1 Q9Y468 2/20 0.38
KDM4E B2RXH2 1/20 0.38
RPS6KB1 P23443 6/20 0.37
AURKA O14965 5/20 0.37
FAAH O00519 7/20 0.36
SLC40A1 Q9NP59 1/20 0.36
PIK3R2 O00459 1/20 0.34
AURKB Q96GD4 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17874765 0.92 PRKDC (0.55) PRKDCKDM4ERPS6KB1AURKAFAAH
SCHEMBL17634672 0.91 PRKDC (0.64) PRKDCL3MBTL1KDM4ERPS6KB1AURKA
SCHEMBL29392854 0.91 PRKDC (0.53) PRKDCKDM4ERPS6KB1AURKAFAAH
SCHEMBL16653844 0.91 PRKDC (0.53) PRKDCKDM4ERPS6KB1AURKAFAAH
SCHEMBL15328651 0.91 PRKDC (0.53) PRKDCKDM4ERPS6KB1AURKAFAAH
SCHEMBL17874684 0.89 PRKDC (0.52) PRKDCKDM4ERPS6KB1AURKAFAAH
SCHEMBL17634566 0.87 PRKDC (0.55) PRKDCL3MBTL1KDM4ERPS6KB1AURKA
SCHEMBL17874734 0.87 PRKDC (0.57) PRKDCKDM4ERPS6KB1AURKAFAAH
SCHEMBL21155543 0.85 PRKDC (0.50) PRKDCL3MBTL1KDM4ERPS6KB1AURKA
SCHEMBL19819867 0.84 PRKDC (0.49) PRKDCL3MBTL1KDM4ERPS6KB1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9376448-B2 DNA-PK inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2016-06-28 US disclosed