SCHEMBL17878632

SCHEMBL17878632

CN(C)C[C@@H](NC(=O)N1Cc2c(NC(=O)c3cccc([N+](=O)[O-])c3)nn(C)c2C1(C)C)c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAK4 O96013 11/20 0.58
CDK2 P24941 4/20 0.58
CDK7 P50613 8/20 0.51
CCNH P51946 8/20 0.51
MNAT1 P51948 8/20 0.51
CCNT1 O60563 1/20 0.49
CCNA2 P20248 1/20 0.49
CDK9 P50750 1/20 0.49
CCNA1 P78396 1/20 0.49
MELK Q14680 2/20 0.46
HIPK4 Q8NE63 1/20 0.46
NTRK1 P04629 2/20 0.42
MAPK1 P28482 2/20 0.42
RPS6KA1 Q15418 2/20 0.42
PLK4 O00444 1/20 0.42
CHEK1 O14757 1/20 0.42
AURKA O14965 1/20 0.42
GAK O14976 1/20 0.42
RPS6KA5 O75582 1/20 0.42
RPS6KA4 O75676 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25947621 0.92 PAK4 (0.60) PAK4CDK2CDK7CCNHMNAT1
SCHEMBL20754495 0.89 PAK4 (0.60) PAK4CDK2CDK7CCNHMNAT1
SCHEMBL20741115 0.85 CDK7 (0.66) PAK4CDK2CDK7CCNHMNAT1
SCHEMBL31687460 0.85 CDK7 (0.66) PAK4CDK2CDK7CCNHMNAT1
SCHEMBL17878639 0.85 CDK7 (0.66) PAK4CDK2CDK7CCNHMNAT1
SCHEMBL25947627 0.84 PAK4 (0.62) PAK4CDK2CDK7CCNHMNAT1
SCHEMBL25947645 0.83 PAK4 (0.58) PAK4CDK2CDK7CCNHMNAT1
SCHEMBL20741165 0.82 CDK7 (0.73) PAK4CDK2CDK7CCNHMNAT1
SCHEMBL20741163 0.82 CDK7 (0.73) PAK4CDK2CDK7CCNHMNAT1
SCHEMBL22924056 0.81 CDK7 (0.57) PAK4CDK2CDK7CCNHMNAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016105528-A2 INHIBITORS OF CYCLIN-DEPENDENT KINASE 7 (CDK7) DANA-FARBER CANCER INSTITUTE, INC. (US) 2016-06-30 WO disclosed