SCHEMBL17893920

SCHEMBL17893920

CCOC(=O)c1cc(OCC)c(I)c(F)c1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.42
CYP3A4 P08684 2/20 0.42
TDP1 Q9NUW8 3/20 0.41
TP53 P04637 2/20 0.41
HTT P42858 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
GAA P10253 1/20 0.41
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA7 P43166 2/20 0.40
CA9 Q16790 2/20 0.40
CA14 Q9ULX7 2/20 0.40
HSD17B10 Q99714 1/20 0.40
DPP4 P27487 2/20 0.39
ALDH1A1 P00352 4/20 0.39
MAPT P10636 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17893884 0.84 TSHR (0.53) TSHRCYP3A4TP53LMNASMN1; SMN2
Water SCHEMBL17895239 0.81 TSHR (0.49) TSHRCYP3A4TP53HTTLMNA
SCHEMBL31171418 0.78 TSHR (0.60) TSHRCYP3A4TDP1LMNASMN1; SMN2
SCHEMBL31171420 0.78 TSHR (0.60) TSHRCYP3A4TDP1LMNASMN1; SMN2
SCHEMBL4510914 0.78 TSHR (0.47) TSHRCYP3A4TDP1TP53HTT
SCHEMBL7592447 0.78 TDP1 (0.48) TSHRTDP1TP53HTTNPSR1
SCHEMBL4501006 0.78 LMNA (0.49) TSHRTDP1TP53HTTNPSR1
SCHEMBL20607773 0.78 TSHR (0.47) TSHRTDP1TP53HTTNPSR1
SCHEMBL29456210 0.78 TSHR (0.47) TSHRTDP1TP53HTTNPSR1
SCHEMBL22533321 0.77 TSHR (0.44) TSHRCYP3A4CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016109221-A1 BTK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2016-07-07 WO disclosed
WO-2016106625-A1 BTK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2016-07-07 WO disclosed