SCHEMBL17895753

SCHEMBL17895753

Cn1c2c(c3cc(Br)ccc31)CCCCC2

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.68
PTGS1 P23219 1/20 0.68
PTGS2 P35354 1/20 0.68
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
MAPT P10636 3/20 0.42
PPARG P37231 1/20 0.42
NCOA2 Q15596 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
KRAS P01116 2/20 0.42
CCNB2 O95067 1/20 0.40
CDK1 P06493 1/20 0.40
CCNB1 P14635 1/20 0.40
GSK3B P49841 1/20 0.40
CCNB3 Q8WWL7 1/20 0.40
BAZ2B Q9UIF8 2/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
KDM4E B2RXH2 2/20 0.39
ALOX15 P16050 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3861613 0.98 ALOX5 (0.65) ALOX5PTGS1PTGS2MEN1KMT2A
SCHEMBL12241734 0.95 ALOX5 (0.60) ALOX5PTGS1PTGS2MEN1KMT2A
SCHEMBL12927722 0.87 ALOX5 (0.55) ALOX5PTGS1PTGS2MAPTKRAS
SCHEMBL9966179 0.85 ALOX5 (0.53) ALOX5PTGS1PTGS2MEN1KMT2A
SCHEMBL15101429 0.80 ALOX5 (0.67) ALOX5PTGS1PTGS2MEN1KMT2A
SCHEMBL1873708 0.79 PTGS1 (0.65) ALOX5PTGS1PTGS2MAPTBAZ2B
SCHEMBL13877233 0.79 ALOX5 (0.65) ALOX5PTGS1PTGS2MEN1KMT2A
SCHEMBL4727325 0.78 MAPT (0.59) PTGS1PTGS2MEN1KMT2AMAPT
SCHEMBL17895804 0.78 PTGS1 (0.68) ALOX5PTGS1PTGS2MEN1KMT2A
SCHEMBL21088049 0.77 HTR2A (0.50) ALOX5PTGS1PTGS2KRASCCNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016109706-A1 FUSED POLYCYCLIC 2-PYRIDINONE ANTIBACTERIAL COMPOUNDS PTC THERAPEUTICS, INC. (US) 2016-07-07 WO disclosed