SCHEMBL17896758

SCHEMBL17896758

COc1ccc2c(c1)nc(-c1cncc(F)c1)n2C1CC1

nearest known ligand 0.65

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 17/20 0.65
CYP11B1 P15538 16/20 0.65
CYP19A1 P11511 3/20 0.65
ADRA2B P18089 2/20 0.65
HTR2B P41595 2/20 0.51
ADRB1 P08588 1/20 0.51
ADRA2A P08913 1/20 0.51
ADRA2C P18825 1/20 0.51
HTR2C P28335 1/20 0.51
PRKACA P17612 1/20 0.50
RPS6KB1 P23443 1/20 0.50
GSK3B P49841 1/20 0.50
ROCK1 Q13464 1/20 0.50
HTR6 P50406 1/20 0.47
PKM P14618 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10175434 0.86 CYP11B2 (0.76) CYP11B2CYP11B1CYP19A1ADRA2BHTR2B
SCHEMBL17896719 0.86 CYP11B2 (0.74) CYP11B2CYP11B1CYP19A1ADRA2BHTR2B
SCHEMBL461190 0.83 CYP11B2 (0.83) CYP11B2CYP11B1CYP19A1HTR2BPRKACA
SCHEMBL10175815 0.82 CYP11B1 (0.48) CYP11B2CYP11B1CYP19A1ADRA2BSMN1; SMN2
SCHEMBL17896674 0.82 CYP11B2 (0.59) CYP11B2CYP11B1CYP19A1ADRA2BHTR2B
SCHEMBL17896644 0.81 CYP11B2 (0.71) CYP11B2CYP11B1CYP19A1ADRA2B
SCHEMBL459353 0.79 CYP11B2 (1.00) CYP11B2CYP11B1CYP19A1ADRA2B
SCHEMBL17896635 0.79 CYP11B2 (0.68) CYP11B2CYP11B1CYP19A1ADRA2BHTR2B
SCHEMBL10175801 0.79 CYP11B1 (1.00) CYP11B2CYP11B1CYP19A1ADRA2B
SCHEMBL17896672 0.79 CYP11B2 (0.64) CYP11B2CYP11B1CYP19A1ADRA2BHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed