SCHEMBL17898663

SCHEMBL17898663

COc1ccnc(C(=O)N[C@H]2CCOC[C@H](Cc3ccccc3)[C@@H](OCC(C)C)[C@H](C)OC2=O)c1OCOC(C)=O

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.32
ABCB1 P08183 2/20 0.30
CTSL P07711 1/20 0.30
CTSS P25774 1/20 0.30
CTSK P43235 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17898818 0.95 RIPK1 (0.32) RIPK1ABCB1
SCHEMBL15366614 0.94 ABCB1 (0.31) ABCB1
SCHEMBL16062585 0.94 ABCB1 (0.31) ABCB1
SCHEMBL16605283 0.92 ABCB1 (0.31) ABCB1
SCHEMBL17898667 0.92 ABCB1 (0.31) ABCB1
SCHEMBL17427098 0.91 RIPK1 (0.35) RIPK1
SCHEMBL19628450 0.90
SCHEMBL17898878 0.89 RIPK1 (0.30) RIPK1
SCHEMBL15373266 0.89 ABCB1 (0.31) ABCB1CTSLCTSSCTSK
SCHEMBL17898670 0.89

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016109290-A1 MACROCYCLIC PICOLINAMIDE COMPOUNDS WITH FUNGICIDAL ACTIVITY DOW AGROSCIENCES LLC (US) 2016-07-07 WO disclosed
WO-2016109291-A1 USE OF MACROCYCLIC PICOLINAMIDES AS FUNGICIDES DOW AGROSCIENCES LLC (US) 2016-07-07 WO disclosed