SCHEMBL17907966

SCHEMBL17907966

CNC1CCc2c(CC(=O)OC)c3cc(OC)ccc3n2C1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 6/20 0.51
AKR1C3 P42330 4/20 0.47
AKR1C2 P52895 1/20 0.46
CNR2 P34972 3/20 0.45
PTGS2 P35354 1/20 0.45
CNR1 P21554 2/20 0.43
PTGDR Q13258 1/20 0.43
MTNR1A P48039 3/20 0.42
MTNR1B P49286 3/20 0.42
TBXA2R P21731 1/20 0.41
HTR6 P50406 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17907923 0.89 PTGDR2 (0.53) PTGDR2AKR1C3AKR1C2CNR2PTGS2
SCHEMBL17907926 0.88 PTGDR2 (0.47) PTGDR2AKR1C3AKR1C2PTGDRTBXA2R
SCHEMBL17907960 0.88 PTGDR2 (0.49) PTGDR2AKR1C3CNR2PTGS2PTGDR
SCHEMBL17907993 0.88 PTGDR2 (0.50) PTGDR2PTGDRTBXA2R
SCHEMBL17907989 0.85 PTGDR2 (0.52) PTGDR2PTGDRTBXA2R
SCHEMBL13278753 0.81 PTGDR2 (0.59) PTGDR2PTGDRTBXA2R
SCHEMBL13278751 0.81 PTGDR2 (0.59) PTGDR2PTGDRTBXA2R
SCHEMBL13278879 0.81 PTGDR2 (0.59) PTGDR2PTGDRTBXA2R
SCHEMBL17907967 0.81 PTGDR2 (0.59) PTGDR2PTGDRTBXA2R
SCHEMBL17907972 0.79 PTGDR2 (0.52) PTGDR2PTGDRTBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697223-B1 7-(HETEROARYL-AMINO)-6,7,8,9-TETRAHYDROPYRIDO[1,2-A]INDOL ACETIC ACID DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2016-07-13 EP disclosed