SCHEMBL1794709

SCHEMBL1794709

Cc1csc(NC(=O)c2nc(C)cc(-c3ccc(F)c(F)c3)c2C)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.53
MAPT P10636 2/20 0.49
NPC1 O15118 8/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
GCK P35557 3/20 0.47
RAB9A P51151 8/20 0.46
KDM4E B2RXH2 2/20 0.45
HSD17B10 Q99714 2/20 0.45
HPGD P15428 2/20 0.44
POLB P06746 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
ALDH1A1 P00352 2/20 0.44
LMNA P02545 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
POLQ O75417 1/20 0.44
TP53 P04637 1/20 0.44
GAA P10253 1/20 0.44
HTT P42858 1/20 0.44
RCE1 Q9Y256 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1797599 0.90 ABL1 (0.53) GRM5MAPTNPC1MEN1KMT2A
SCHEMBL1796743 0.89 GRM5 (0.63) GRM5MAPTNPC1MEN1KMT2A
SCHEMBL1797295 0.85 GRM5 (0.53) GRM5MAPTNPC1MEN1KMT2A
SCHEMBL1794178 0.84 GRM5 (0.54) GRM5MAPTNPC1MEN1KMT2A
SCHEMBL1794339 0.83 GRM5 (0.45) GRM5NPC1MEN1KMT2ARAB9A
SCHEMBL1794766 0.81 GRM5 (0.49) GRM5MAPTNPC1MEN1KMT2A
SCHEMBL1796425 0.81 SMARCA2 (0.57) GRM5MAPTNPC1MEN1KMT2A
SCHEMBL1796910 0.81 GRM5 (0.52) GRM5MAPTNPC1MEN1KMT2A
SCHEMBL1797024 0.80 GRM5 (0.54) GRM5MAPTNPC1MEN1KMT2A
SCHEMBL1798452 0.80 GRM5 (0.52) GRM5MAPTNPC1GCKRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7951824-B2 4-aryl-pyridine-2-carboxyamide derivatives HOFFMAN-LA ROCHE INC. (US) 2011-05-31 US claimed
US-7951824-B2 4-aryl-pyridine-2-carboxyamide derivatives HOFFMAN-LA ROCHE INC. (US) 2011-05-31 US disclosed