SCHEMBL1795189

SCHEMBL1795189

Cc1cccc(NC(=O)c2cc(-c3cccnc3)cc(C)n2)n1

nearest known ligand 0.67

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 7/20 0.60
CYP1A2 P05177 2/20 0.57
CYP2C9 P11712 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1794792 0.91 GRM5 (0.50) GRM5CYP1A2CYP2C9
SCHEMBL1793909 0.86 KMT2A (0.53) GRM5CYP1A2CYP2C9
SCHEMBL30761182 0.84 GRM5 (0.56) GRM5CYP1A2CYP2C9
SCHEMBL3864114 0.83 GRM5 (0.66) GRM5
SCHEMBL1796059 0.83 SMN1; SMN2 (0.58) CYP1A2CYP2C9
SCHEMBL1796217 0.83 IRAK4 (0.47) GRM5
SCHEMBL1795519 0.82 NPC1 (0.47) GRM5
SCHEMBL15890661 0.81 CYP1A2 (0.80) GRM5CYP1A2CYP2C9
SCHEMBL5029221 0.81 GRM5 (0.70) GRM5
SCHEMBL1796357 0.80 GRM5 (0.68) GRM5CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7951824-B2 4-aryl-pyridine-2-carboxyamide derivatives HOFFMAN-LA ROCHE INC. (US) 2011-05-31 US claimed
US-7951824-B2 4-aryl-pyridine-2-carboxyamide derivatives HOFFMAN-LA ROCHE INC. (US) 2011-05-31 US disclosed