SCHEMBL17957098

SCHEMBL17957098

O=C(c1ccc(F)cc1F)N1CCC(N2C[C](n3cc(-c4ncnc5[nH]ccc45)cn3)C2)CC1

nearest known ligand 0.68

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 20/20 0.68
JAK1 P23458 10/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17957111 0.94 JAK2 (0.68) JAK2JAK1
SCHEMBL14563469 0.92 JAK2 (0.68) JAK2JAK1
SCHEMBL14563579 0.91 JAK2 (0.70) JAK2JAK1
SCHEMBL14563758 0.91 JAK2 (0.60) JAK2JAK1
SCHEMBL17387462 0.91 JAK2 (0.68) JAK2JAK1
SCHEMBL14563568 0.90 JAK2 (0.57) JAK2JAK1
SCHEMBL14563398 0.90 JAK2 (0.68) JAK2JAK1
SCHEMBL14563756 0.89 JAK2 (0.68) JAK2JAK1
SCHEMBL14563900 0.89 JAK2 (0.57) JAK2JAK1
SCHEMBL17387451 0.89 JAK2 (0.67) JAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3050882-A1 PIPERIDIN-4-YL AZETIDINE DERIVATIVES AS JAK1 INHIBITORS Incyte Holdings Corporation (US) 2016-08-03 EP claimed
EP-4400172-A2 PIPERIDIN-4-YL AZETIDINE DERIVATIVES AS JAK1 INHIBITORS Incyte Holdings Corporation (US) 2024-07-17 EP disclosed
EP-3354652-A1 PIPERIDIN-4-YL AZETIDINE DERIVATIVES AS JAK1 INHIBITORS Incyte Holdings Corporation (US) 2018-08-01 EP disclosed