SCHEMBL17957258

SCHEMBL17957258

O=C(CCCc1nc(OC(=O)O)c(NC(=O)Nc2ccc(Cl)cc2)[nH]1)Nc1ccc2[nH]nnc2c1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 5/20 0.38
NTRK2 Q16620 3/20 0.38
MAPT P10636 1/20 0.37
ALDH1A1 P00352 2/20 0.36
POLB P06746 1/20 0.36
PARP1 P09874 2/20 0.36
NPY5R Q15761 1/20 0.34
ROCK2 O75116 1/20 0.34
ROCK1 Q13464 1/20 0.34
MMP2 P08253 1/20 0.34
MMP13 P45452 1/20 0.34
TNKS O95271 1/20 0.34
PARP2 Q9UGN5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17957276 0.90 MCHR1 (0.40) NTRK1NTRK2ALDH1A1PARP1
SCHEMBL2815670 0.88 NTRK1 (0.40) NTRK1NTRK2MAPTALDH1A1POLB
SCHEMBL17957241 0.88 MAPT (0.39) NTRK1NTRK2MAPTALDH1A1ROCK2
SCHEMBL17957242 0.86 ROCK2 (0.50) ROCK2ROCK1
SCHEMBL13133022 0.86 PARP1 (0.41) NTRK1NTRK2MAPTALDH1A1POLB
SCHEMBL17957277 0.85 NTRK1 (0.39) NTRK1NTRK2MAPTALDH1A1POLB
SCHEMBL17957281 0.85 MCHR1 (0.43) NTRK1NTRK2MAPTALDH1A1
SCHEMBL2814887 0.81 MAPT (0.41) NTRK1NTRK2MAPTALDH1A1PARP1
SCHEMBL2815410 0.78 MCHR1 (0.42) NTRK1NTRK2ALDH1A1PARP1
SCHEMBL17957284 0.78 NTRK1 (0.42) NTRK1NTRK2ALDH1A1PARP1MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2193122-B1 IMIDAZOLE DERIVATIVES MERCK PATENT GMBH (DE) 2016-08-03 EP claimed
EP-2193122-B1 IMIDAZOLE DERIVATIVES MERCK PATENT GMBH (DE) 2016-08-03 EP disclosed