SCHEMBL1796559

SCHEMBL1796559

Cc1cc(-c2ccccn2)cc(C(=O)Nc2nc(C)cs2)n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.56
RAB9A P51151 6/20 0.56
GRM5 P41594 4/20 0.54
KDM4E B2RXH2 3/20 0.53
GAA P10253 2/20 0.53
KMT2A Q03164 3/20 0.53
GCK P35557 1/20 0.53
CASP3 P42574 1/20 0.53
SENP8 Q96LD8 1/20 0.53
SENP7 Q9BQF6 1/20 0.53
SENP6 Q9GZR1 1/20 0.53
ADORA3 P0DMS8 3/20 0.53
KDM4A O75164 1/20 0.52
KDM4B O94953 1/20 0.52
KDM5B Q9UGL1 1/20 0.52
L3MBTL1 Q9Y468 3/20 0.51
HTT P42858 3/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
HSP90AA1 P07900 1/20 0.51
MEN1 O00255 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1795585 0.84 GRM5 (0.52) NPC1RAB9AGRM5KDM4EGAA
SCHEMBL1795424 0.84 NPC1 (0.70) NPC1RAB9AGRM5KDM4EGAA
SCHEMBL12258301 0.84 NPC1 (0.71) NPC1RAB9AGRM5KDM4EGAA
SCHEMBL1796144 0.83 GRM5 (0.58) NPC1RAB9AGRM5KDM4EGAA
SCHEMBL1794974 0.83 GRM5 (0.53) NPC1RAB9AGRM5KDM4EGAA
SCHEMBL29074201 0.82 NPC1 (0.60) NPC1RAB9AGRM5KDM4EGAA
SCHEMBL1793529 0.81 NPC1 (0.56) NPC1RAB9AGRM5KDM4EGAA
SCHEMBL1797781 0.81 SMARCA2 (0.61) NPC1RAB9AGRM5KDM4EGAA
SCHEMBL1798244 0.80 GRM5 (0.60) NPC1RAB9AGRM5KDM4EGAA
SCHEMBL1796021 0.80 GRM5 (0.54) NPC1RAB9AGRM5KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7951824-B2 4-aryl-pyridine-2-carboxyamide derivatives HOFFMAN-LA ROCHE INC. (US) 2011-05-31 US claimed
US-7951824-B2 4-aryl-pyridine-2-carboxyamide derivatives HOFFMAN-LA ROCHE INC. (US) 2011-05-31 US disclosed