SCHEMBL17969745

SCHEMBL17969745

Fc1ccc(Cl)c(CN2CCNc3c2c2c(-c4ccc(N5CCOCC5)cc4)n3-2)c1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
CYP2A13 Q16696 2/20 0.35
CNR2 P34972 1/20 0.35
PLK4 O00444 1/20 0.35
JAK2 O60674 1/20 0.35
PRKD3 O94806 1/20 0.35
MAP4K4 O95819 1/20 0.35
ABL1 P00519 1/20 0.35
LCK P06239 1/20 0.35
CSF1R P07333 1/20 0.35
RET P07949 1/20 0.35
MET P08581 1/20 0.35
ROS1 P08922 1/20 0.35
FGFR1 P11362 1/20 0.35
SRC P12931 1/20 0.35
FER P16591 1/20 0.35
FGFR3 P22607 1/20 0.35
LTK P29376 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17969728 0.79 ALK (0.49) CNR2PLK4JAK2PRKD3MAP4K4
SCHEMBL20859359 0.77 KDM4E (0.39) KDM4EALDH1A1HPGDCYP2A13CNR2
SCHEMBL17918716 0.75 ALK (0.46) KDM4EALDH1A1HPGDCYP2A13CNR2
SCHEMBL16615279 0.74 HDAC1 (0.33) PLK4JAK2PRKD3MAP4K4ABL1
SCHEMBL17969742 0.71 KDM4E (0.35) KDM4EALDH1A1HPGDCYP2A13MAPT
SCHEMBL16615200 0.71 CHRM1 (0.45) JAK2
SCHEMBL16615167 0.70 MAP4K3 (0.31) JAK2
SCHEMBL16615312 0.70 NR1H4 (0.36)
SCHEMBL17918740 0.70 ALK (0.40) KDM4EALDH1A1HPGDCYP2A13PLK4
SCHEMBL1601010 0.69 ALK (0.67) KDM4EALDH1A1HPGDPLK4JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3050884-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES Limited Liability Company "National Pharmaceutical (RU) 2016-08-03 EP disclosed