SCHEMBL17970569

SCHEMBL17970569

CCCc1cc(C)c(CNN=N)c(=O)[nH]1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
HPGD P15428 3/20 0.38
KDM4E B2RXH2 3/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
HSD17B10 Q99714 2/20 0.37
CYP1A2 P05177 1/20 0.37
TSHR P16473 3/20 0.36
MPO P05164 1/20 0.36
TPO P07202 1/20 0.36
LPO P22079 1/20 0.36
CYP2C19 P33261 1/20 0.36
TAS2R38 P59533 1/20 0.36
ADORA1 P30542 2/20 0.36
ADORA2A P29274 1/20 0.36
PKM P14618 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
RAB9A P51151 1/20 0.33
MAPT P10636 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17970510 0.80 EZH2 (0.42) KDM4EPKMEZH2EEDRBBP4
SCHEMBL17970524 0.77 EED (0.45) ALDH1A1HPGDKDM4EHSD17B10PKM
SCHEMBL1695068 0.75 TSHR (0.42) ALDH1A1HPGDKDM4EGLAGAA
SCHEMBL17970490 0.71 EZH2 (0.35) ALDH1A1HPGDKDM4EGLAGAA
SCHEMBL18560159 0.71 TSHR (0.47) ALDH1A1HPGDKDM4EGLAGAA
SCHEMBL1694783 0.68 KDM4E (0.64) ALDH1A1HPGDKDM4EGLAGAA
SCHEMBL21156095 0.68 EZH2 (0.41) ALDH1A1HPGDKDM4EHSD17B10PKM
SCHEMBL17970362 0.67 KDM4E (0.35) KDM4EGAAPKMEZH2EED
Trifluoroacetic Acid SCHEMBL1695078 0.66 KDM4E (0.41) ALDH1A1HPGDKDM4EGLAGAA
SCHEMBL12570733 0.63 MPO (0.44) ALDH1A1HPGDKDM4EGLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2773754-B1 Compounds for use in the treatment of T-cell mediated diseases GLAXOSMITHKLINE IP NO 2 LTD (GB) 2016-08-03 EP disclosed