SCHEMBL18009377

SCHEMBL18009377

O=C1CNC(=O)[C@H](COC(=O)/C=C/C(=O)OCc2ccccc2)N1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 5/20 0.55
GLA P06280 1/20 0.46
LMNA P02545 1/20 0.46
AKR1B10 O60218 2/20 0.43
AKR1B1 P15121 2/20 0.43
CA12 O43570 2/20 0.43
CA4 P22748 2/20 0.43
CA6 P23280 2/20 0.43
CA5A P35218 2/20 0.43
CA7 P43166 2/20 0.43
CA9 Q16790 2/20 0.43
CA14 Q9ULX7 2/20 0.43
CA5B Q9Y2D0 2/20 0.43
TTR P02766 1/20 0.40
NAAA Q02083 1/20 0.40
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
OPRM1 P35372 2/20 0.38
OPRD1 P41143 2/20 0.38
OPRK1 P41145 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18009369 0.87 HCAR2 (0.37) HCAR2GLAALDH1A1OPRM1OPRD1
SCHEMBL18007432 0.86 HRH3 (0.34) HCAR2
SCHEMBL18007431 0.86 HRH3 (0.34) HCAR2
SCHEMBL18014853 0.83 HCAR2 (0.54) HCAR2GLALMNAAKR1B10AKR1B1
SCHEMBL18015918 0.81 HCAR2 (0.58) HCAR2GLALMNAAKR1B10AKR1B1
SCHEMBL16088 0.81 LMNA (0.50) GLALMNAOPRM1OPRD1OPRK1
SCHEMBL16543 0.81 LMNA (0.50) GLALMNAOPRM1OPRD1OPRK1
SCHEMBL4840306 0.81 LMNA (0.50) GLALMNAOPRM1OPRD1OPRK1
SCHEMBL31377175 0.80 GLA (0.67) GLANAAAALDH1A1DDB1CRBN
SCHEMBL18009220 0.80 HCAR2 (0.36) HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016127186-A1 FUMARATE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND METHODS OF USE NGUYEN MARK QUANG (US) 2016-08-11 WO disclosed