SCHEMBL18018564

SCHEMBL18018564

O=C(NCc1cc(-c2cnc(C(F)(F)F)nc2)cnc1C1CC1)[C@@H]1C[C@@H](F)CN1S(=O)(=O)c1ccc(F)cc1

nearest known ligand 0.83

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 20/20 0.83

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16647857 0.91 TRPA1 (1.00) TRPA1
SCHEMBL16634892 0.88 TRPA1 (1.00) TRPA1
SCHEMBL18018464 0.88 TRPA1 (0.83) TRPA1
SCHEMBL18017850 0.88 TRPA1 (0.84) TRPA1
SCHEMBL16647887 0.87 TRPA1 (1.00) TRPA1
SCHEMBL16634891 0.85 TRPA1 (0.83) TRPA1
SCHEMBL18017847 0.85 TRPA1 (0.82) TRPA1
SCHEMBL16635043 0.85 TRPA1 (1.00) TRPA1
SCHEMBL18047620 0.85 TRPA1 (0.75) TRPA1
SCHEMBL18018075 0.85 TRPA1 (0.75) TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016128529-A1 1-(HET)ARYLSULFONYL-(PYRROLIDINE OR PIPERIDINE)-2-CARBOXAMIDE DERIVATIVES AND THEIR USE AS TRPA1 ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2016-08-18 WO disclosed