SCHEMBL18025331

SCHEMBL18025331

Cc1ccc(NC(=O)Nc2cc(CF)cc(C(F)(F)F)c2)cc1OCCN1CCNCC1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.46
HTR2A P28223 4/20 0.46
HTR2C P28335 4/20 0.46
EPHX2 P34913 3/20 0.45
RAF1 P04049 1/20 0.45
QPCT Q16769 1/20 0.45
KDR P35968 3/20 0.42
BRAF P15056 3/20 0.42
MCHR1 Q99705 2/20 0.41
RXFP1 Q9HBX9 2/20 0.41
ERN1 O75460 1/20 0.40
MAPK14 Q16539 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18196958 0.93 IDH1 (0.50) IDH1HTR2AHTR2CEPHX2RAF1
Hydrochloric Acid SCHEMBL2682150 0.92 RAF1 (0.49) IDH1HTR2AHTR2CEPHX2RAF1
SCHEMBL2682353 0.82 EPHX2 (0.64) HTR2AHTR2CEPHX2RAF1BRAF
SCHEMBL4554237 0.81 BRAF (0.61) HTR2AHTR2CEPHX2RAF1QPCT
SCHEMBL18196957 0.79 RAF1 (0.48) IDH1HTR2AHTR2CRAF1MCHR1
SCHEMBL10220711 0.79 HTR2A (0.56) HTR2AHTR2CEPHX2QPCTKDR
Hydrochloric Acid SCHEMBL2681808 0.78 HTR2A (0.55) HTR2AHTR2CEPHX2QPCTKDR
SCHEMBL11008302 0.74 PSEN1 (0.48) IDH1HTR2AHTR2CEPHX2RAF1
SCHEMBL18025318 0.74 CA12 (0.47) IDH1EPHX2KDR
SCHEMBL6874112 0.73 LMNA (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9421211-B2 N,N′-diarylurea compounds and N,N′-diarylthiourea compounds as inhibitors of translation initiation PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2016-08-23 US disclosed