SCHEMBL18030076

SCHEMBL18030076

CCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O

nearest known ligand 0.67

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 6/20 0.67
NOD1 Q9Y239 2/20 0.61
GLP1R P43220 8/20 0.60
EPHX2 P34913 4/20 0.56
RIMKLA Q8IXN7 1/20 0.54
NAALAD2 Q9Y3Q0 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12836737 1.00 FOLH1 (0.67) FOLH1NOD1GLP1REPHX2RIMKLA
SCHEMBL22237179 1.00 FOLH1 (0.67) FOLH1NOD1GLP1REPHX2RIMKLA
SCHEMBL21417883 1.00 FOLH1 (0.67) FOLH1NOD1GLP1REPHX2RIMKLA
SCHEMBL15003787 1.00 FOLH1 (0.67) FOLH1NOD1GLP1REPHX2RIMKLA
SCHEMBL20018407 1.00 FOLH1 (0.67) FOLH1NOD1GLP1REPHX2RIMKLA
SCHEMBL20018413 1.00 FOLH1 (0.67) FOLH1NOD1GLP1REPHX2RIMKLA
SCHEMBL18059393 0.99 FOLH1 (0.69) FOLH1NOD1GLP1REPHX2RIMKLA
SCHEMBL16645331 0.97 NOD1 (0.65) FOLH1NOD1GLP1REPHX2
SCHEMBL15003786 0.97 NOD1 (0.65) FOLH1NOD1GLP1REPHX2
SCHEMBL23252356 0.97 FOLH1 (0.67) FOLH1NOD1GLP1REPHX2RIMKLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3545978-B1 TRIAZINE BASED RADIOPHARMACEUTICALS AND RADIOIMAGING AGENTS MOLECULAR INSIGHT PHARM INC (US) 2021-09-08 EP disclosed
EP-3545978-A1 TRIAZINE BASED RADIOPHARMACEUTICALS AND RADIOIMAGING AGENTS Molecular Insight Pharmaceuticals, Inc. (US) 2019-10-02 EP disclosed
EP-3300746-B1 TRIAZINE BASED RADIOPHARMACEUTICALS AND RADIOIMAGING AGENTS MOLECULAR INSIGHT PHARM INC (US) 2019-05-15 EP disclosed
EP-3300746-A1 TRIAZINE BASED RADIOPHARMACEUTICALS AND RADIOIMAGING AGENTS Molecular Insight Pharmaceuticals, Inc. (US) 2018-04-04 EP disclosed
EP-2943227-B1 TRIAZINE BASED RADIOPHARMACEUTICALS AND RADIOIMAGING AGENTS MOLECULAR INSIGHT PHARM INC (US) 2017-09-20 EP disclosed
EP-2389361-B1 TECHNETIUM- AND RHENIUM-BIS(HETEROARYL) COMPLEXES AND METHODS OF USE THEREOF FOR INHIBITING PSMA MOLECULAR INSIGHT PHARM INC (US) 2016-08-24 EP disclosed