SCHEMBL1804004

SCHEMBL1804004

CC(C)(C)c1ccc(COc2ccc(Cn3cc(-c4cccnc4N)nn3)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 7/20 0.55
HSP90AB1 P08238 7/20 0.55
APP P05067 1/20 0.42
CCNK O75909 1/20 0.42
CDK12 Q9NYV4 1/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
PSEN1 P49768 1/20 0.41
PSEN2 P49810 1/20 0.41
KCNH2 Q12809 1/20 0.41
APH1B Q8WW43 1/20 0.41
NCSTN Q92542 1/20 0.41
APH1A Q96BI3 1/20 0.41
PSENEN Q9NZ42 1/20 0.41
CYP19A1 P11511 3/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
TP53 P04637 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NR4A2 P43354 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1808527 0.90 NPC1 (0.53) HSP90AA1HSP90AB1CCNKCDK12NPC1
SCHEMBL1734185 0.89 CYP19A1 (0.51) CCNKCDK12CYP19A1MEN1KMT2A
SCHEMBL1813784 0.88 CYP19A1 (0.52) CCNKCDK12NPC1RAB9ACYP19A1
SCHEMBL1816497 0.88 TEK (0.43) CCNKCDK12NPC1RAB9ACYP19A1
SCHEMBL1806051 0.87 EPHB4 (0.45) CCNKCDK12NPC1RAB9ACYP19A1
SCHEMBL1812647 0.85 HSP90AA1 (0.45) HSP90AA1HSP90AB1CCNKCDK12NPC1
SCHEMBL1816014 0.84 CCNK (0.47) HSP90AA1HSP90AB1CCNKCDK12NPC1
SCHEMBL1805271 0.84 CCNK (0.56) HSP90AA1HSP90AB1CCNKCDK12NPC1
SCHEMBL1809812 0.83 CD74 (0.53) CCNKCDK12NPC1RAB9ACYP19A1
SCHEMBL1806532 0.83 KDR (0.47) CCNKCDK12NPC1RAB9ACYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011051198-A2 PYRIDINE DERIVATIVES AS AGRICULTURAL PESTICIDES BAYER CROPSCIENCE AG (DE) 2011-05-05 WO claimed
WO-2011051198-A2 PYRIDINE DERIVATIVES AS AGRICULTURAL PESTICIDES BAYER CROPSCIENCE AG (DE) 2011-05-05 WO disclosed