SCHEMBL18052175

SCHEMBL18052175

CC(C)(C)C(=O)Nc1cc(N(N)C2CCN(C(=O)OCc3ccccc3)CC2)c(Br)cn1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
GRIN2B Q13224 9/20 0.43
CYP2D6 P10635 4/20 0.43
CYP2C9 P11712 4/20 0.43
CYP3A4 P08684 3/20 0.43
CYP2C19 P33261 1/20 0.43
HTT P42858 1/20 0.42
MAPK1 P28482 1/20 0.41
USP30 Q70CQ3 1/20 0.41
CA2 P00918 1/20 0.41
GPR119 Q8TDV5 1/20 0.40
LNPEP Q9UIQ6 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL617560 0.82 GRIN2B (0.45) SMN1; SMN2NPC1RAB9AGRIN2BCYP2D6
SCHEMBL617505 0.81 GRIN2B (0.57) GRIN2BCYP2D6CYP2C9CYP3A4CA2
SCHEMBL620312 0.74 GRIN2B (0.57) GRIN2BCYP2D6CYP2C9CYP3A4
SCHEMBL3166460 0.72 SMN1; SMN2 (0.47) SMN1; SMN2NPC1RAB9AGRIN2BCYP2D6
SCHEMBL12124917 0.70 GRIN2B (0.45) SMN1; SMN2NPC1RAB9AGRIN2BCYP2D6
SCHEMBL3933073 0.69 SMN1; SMN2 (0.57) SMN1; SMN2NPC1RAB9AGRIN2BCYP2D6
SCHEMBL8550410 0.69 SMN1; SMN2 (0.66) SMN1; SMN2NPC1RAB9AGRIN2BCYP2D6
SCHEMBL13547205 0.68 SMN1; SMN2 (0.55) SMN1; SMN2NPC1RAB9AGRIN2BCYP2D6
SCHEMBL23706353 0.68 SMN1; SMN2 (0.68) SMN1; SMN2NPC1RAB9AGRIN2BCYP2D6
SCHEMBL20135084 0.67 SMN1; SMN2 (0.58) SMN1; SMN2NPC1RAB9AGRIN2BCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2197874-B1 PYRAZIN-2-YL-PYRIDIN-2-YL-AMINE AND PYRAZIN-2-YL-PYRIMIDIN-4-YL-AMINE COMPOUNDS AND THEIR USE CANCER REC TECH LTD (GB) 2016-08-31 EP disclosed