SCHEMBL18059809

SCHEMBL18059809

C(=C/c1ccccc1)\Cc1cccnc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.58
CYP11B2 P19099 1/20 0.58
TBXAS1 P24557 3/20 0.48
G6PC1 P35575 1/20 0.46
LTA4H P09960 1/20 0.46
CYP2D6 P10635 3/20 0.45
CYP1A2 P05177 3/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 2/20 0.45
CYP1A1 P04798 1/20 0.45
CYP1B1 Q16678 1/20 0.45
CHRNB2 P17787 1/20 0.45
CHRNB4 P30926 1/20 0.45
CHRNA3 P32297 1/20 0.45
CHRNA7 P36544 1/20 0.45
CHRNA4 P43681 1/20 0.45
MEN1 O00255 1/20 0.45
ALOX15 P16050 1/20 0.45
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18059810 1.00 CYP11B1 (0.58) CYP11B1CYP11B2TBXAS1G6PC1LTA4H
Piperazine SCHEMBL28139495 0.91 CYP11B1 (0.49) CYP11B1CYP11B2TBXAS1G6PC1LTA4H
SCHEMBL24384517 0.81 CYP11B1 (0.57) CYP11B1CYP11B2TBXAS1CYP2D6CYP1A2
SCHEMBL9584872 0.81 CYP11B2 (0.52) CYP11B1CYP11B2G6PC1LTA4HCYP2D6
SCHEMBL6960280 0.81 CYP3A4 (0.52) CYP11B1CYP11B2TBXAS1CYP2D6CYP1A2
SCHEMBL6958821 0.81 CYP3A4 (0.52) CYP11B1CYP11B2TBXAS1CYP2D6CYP1A2
SCHEMBL6958816 0.81 CYP3A4 (0.52) CYP11B1CYP11B2TBXAS1CYP2D6CYP1A2
SCHEMBL4256257 0.80 MAOB (0.67) LTA4HCYP3A4MEN1ALOX15KMT2A
SCHEMBL163963 0.80 MAOB (0.67) LTA4HCYP3A4MEN1ALOX15KMT2A
SCHEMBL1892917 0.80 MAOB (0.67) LTA4HCYP3A4MEN1ALOX15KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016146689-A1 ORGANOZINC REAGENTS AND PROCESSES FOR PREPARING AND USING THE SAME LUDWIG-MAXIMILIANS-UNIVERSITÄT MÜNCHEN (DE) 2016-09-22 WO disclosed
EP-3070083-A1 Organozinc reagents and processes for preparing and using the same Ludwig-Maximilians-Universität München (DE) 2016-09-21 EP disclosed
EP-3070083-A1 Organozinc reagents and processes for preparing and using the same Ludwig-Maximilians-Universität München (DE) 2016-09-21 EP disclosed