SCHEMBL18069130

SCHEMBL18069130

Cc1cccc2[nH]cc(Br)c12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 3/20 0.58
CYP2A6 P11509 1/20 0.46
HTR2A P28223 2/20 0.44
ATM Q13315 1/20 0.42
ALDH1A1 P00352 1/20 0.39
SLC6A4 P31645 1/20 0.38
AHR P35869 1/20 0.36
CLK1 P49759 1/20 0.36
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
FFAR1 O14842 1/20 0.36
ALKBH5 Q6P6C2 1/20 0.35
FTO Q9C0B1 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
NPC1 O15118 1/20 0.35
KIF11 P52732 1/20 0.34
PARP1 P09874 1/20 0.34
MAPK1 P28482 1/20 0.34
MAP2K4 P45985 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3614670 0.83 CYP2A6 (0.55) GPR84CYP2A6HTR2AATMALDH1A1
SCHEMBL31663257 0.83 CYP2A6 (0.55) GPR84CYP2A6HTR2AATMALDH1A1
SCHEMBL28973447 0.80 CYP2A6 (0.60) GPR84CYP2A6HTR2ASLC6A4AHR
SCHEMBL1224614 0.80 GPR84 (0.64) GPR84CYP2A6HTR2AATMALDH1A1
SCHEMBL30552280 0.80 GPR84 (0.64) GPR84CYP2A6HTR2AATMALDH1A1
SCHEMBL17308781 0.75 GPR84 (0.58) GPR84HTR2AATMSLC6A4FFAR1
SCHEMBL5924727 0.75 GPR84 (0.58) GPR84CYP2A6HTR2AATMFFAR1
SCHEMBL20905344 0.75 CYP2A6 (0.46) GPR84CYP2A6HTR2AALDH1A1SLC6A4
SCHEMBL1224297 0.75 GPR84 (0.58) GPR84HTR2AATMSLC6A4FFAR1
SCHEMBL4587369 0.75 GPR84 (0.58) GPR84CYP2A6SLC6A4AHRCLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016144702-A1 LYSYL OXIDASE-LIKE 2 INHIBITORS AND USES THEREOF PHARMAKEA, INC. (US) 2016-09-15 WO disclosed