SCHEMBL18075876

SCHEMBL18075876

Cc1c(-c2nc(C(=O)O)nn2-c2ccc(C#N)cc2)cn2nc(NC(=O)CCCN(C)C)nc2c1-c1cccc(C(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35
MALT1 Q9UDY8 1/20 0.35
ELANE P08246 6/20 0.35
TP53 P04637 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CTSK P43235 2/20 0.34
ADORA2A P29274 1/20 0.34
RXFP1 Q9HBX9 1/20 0.33
TRPV4 Q9HBA0 1/20 0.33
MAPT P10636 1/20 0.32
MGAT2 Q10469 1/20 0.32
CCR2 P41597 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18076215 0.94 MALT1 (0.37) KMT2AALDH1A1NPSR1KDM4EHPGD
SCHEMBL15425551 0.91 KMT2A (0.40) KMT2AALDH1A1NPSR1KDM4EHPGD
SCHEMBL15412416 0.89 MALT1 (0.35) MALT1ELANECTSKADORA2ARXFP1
Formic Acid SCHEMBL15412152 0.89 KMT2A (0.38) KMT2AALDH1A1NPSR1KDM4EHPGD
Formic Acid SCHEMBL15412150 0.89 KMT2A (0.37) KMT2AALDH1A1NPSR1KDM4EHPGD
SCHEMBL18043803 0.88 KMT2A (0.45) KMT2AALDH1A1NPSR1KDM4EHPGD
SCHEMBL15412357 0.88 ELANE (0.44) MALT1ELANECTSKADORA2ATRPV4
SCHEMBL15412140 0.86 MALT1 (0.36) MALT1ELANECTSKADORA2AMGAT2
SCHEMBL15425558 0.85 MALT1 (0.37) KMT2AALDH1A1NPSR1KDM4EHPGD
Bromide SCHEMBL15412068 0.85 MALT1 (0.36) KMT2AALDH1A1NPSR1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2872509-B1 INHIBITION OF ENZYMES CHIESI FARMA SPA (IT) 2016-09-14 EP disclosed