SCHEMBL1809475

SCHEMBL1809475

Cc1ccc2ncc(Br)nc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.50
ABL1 P00519 1/20 0.49
RET P07949 1/20 0.49
KDR P35968 1/20 0.49
CDK7 P50613 1/20 0.49
CDK5 Q00535 1/20 0.49
PRKAA1 Q13131 1/20 0.49
AURKB Q96GD4 1/20 0.49
CLK4 Q9HAZ1 1/20 0.49
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 3/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MAPT P10636 4/20 0.42
TDP1 Q9NUW8 1/20 0.42
CYP1A2 P05177 3/20 0.41
MAPK1 P28482 2/20 0.40
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
IKBKB O14920 1/20 0.38
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14330664 0.92 NQO2 (0.50) NQO2ABL1RETKDRCDK7
SCHEMBL8344116 0.79 CYP1A2 (0.54) NQO2CDK5ALDH1A1KDM4EL3MBTL1
SCHEMBL30578800 0.79 CYP1A2 (0.54) NQO2CDK5ALDH1A1KDM4EL3MBTL1
SCHEMBL29639029 0.79 CYP1A2 (0.54) NQO2CDK5ALDH1A1KDM4EL3MBTL1
SCHEMBL26919701 0.79 HTT (0.44) ABL1RETKDRCDK7CDK5
SCHEMBL26790744 0.77 ALDH1A1 (0.47) NQO2ALDH1A1KDM4EL3MBTL1MAPT
SCHEMBL28286272 0.77 ALDH1A1 (0.57) NQO2ABL1RETKDRCDK7
SCHEMBL6845013 0.76 BACE1 (0.55) NQO2ALDH1A1KDM4EL3MBTL1MAPT
SCHEMBL19001534 0.76 NQO2 (0.50) NQO2ALDH1A1KDM4EL3MBTL1MAPT
SCHEMBL1256925 0.76 FGFR3 (0.46) KDRALDH1A1KDM4EMAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2321296-A1 SUBSTITUTED 5-AMINOPYRAZOLES AND USE THEREOF Bayer Schering Pharma Aktiengesellschaft (DE) 2011-05-18 EP disclosed
WO-2010020363-A1 SUBSTITUTED 5-AMINOPYRAZOLES AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-02-25 WO disclosed