Thiophene Carboxylic Acid

Thiophene Carboxylic Acid

SCHEMBL18112600

O=C(Cl)c1cccs1.O=C(O)c1cccs1

nearest known ligand 0.79

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.79
CES2 O00748 2/20 0.56
CES1 P23141 2/20 0.56
HPGDS O60760 1/20 0.52
GSK3B P49841 1/20 0.52
LMNA P02545 3/20 0.52
ALOX15 P16050 1/20 0.52
MEN1 O00255 4/20 0.50
KMT2A Q03164 4/20 0.50
RAB9A P51151 4/20 0.50
NPC1 O15118 3/20 0.50
ALDH1A1 P00352 2/20 0.50
POLB P06746 1/20 0.50
HDAC1 Q13547 1/20 0.50
ERCC5 P28715 1/20 0.47
FEN1 P39748 1/20 0.47
TDP1 Q9NUW8 1/20 0.46
HPGD P15428 3/20 0.44
TP53 P04637 1/20 0.44
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Thiophene Carboxylic Acid SCHEMBL27932787 0.91 DAO (0.86) DAOCES2CES1HPGDSGSK3B
SCHEMBL1813 0.91
Hydrochloric Acid SCHEMBL28208472 0.89
Thiophene Carboxylic Acid SCHEMBL7062244 0.89 DAO (1.00) DAOCES2CES1HPGDSGSK3B
Thiophene Carboxylic Acid SCHEMBL27774764 0.89 DAO (1.00) DAOCES2CES1HPGDSGSK3B
Thiophene Carboxylic Acid SCHEMBL83000 0.89
Thiophene Carboxylic Acid SCHEMBL5287669 0.87 DAO (0.95) DAOCES2CES1HPGDSGSK3B
Thiophene Carboxylic Acid SCHEMBL1814 0.87
Thiophene Carboxylic Acid SCHEMBL20895852 0.87
Thiophene Carboxylic Acid SCHEMBL11452200 0.87

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3433242-A1 PROCESSES FOR THE PREPARATION OF HETEROARYL CARBOXYLIC ACIDS Monsanto Technology LLC (US) 2019-01-30 EP disclosed
EP-3277275-A1 PROCESSES FOR THE PREPARATION OF 2-THIOPHENECARBONYL CHLORIDE Monsanto Technology LLC (US) 2018-02-07 EP disclosed
WO-2017165356-A1 PROCESSES FOR THE PREPARATION OF HETEROARYL CARBOXYLIC ACIDS MONSANTO TECHNOLOGY LLC (US) 2017-09-28 WO disclosed
WO-2016161063-A1 PROCESSES FOR THE PREPARATION OF 2-THIOPHENECARBONYL CHLORIDE MONSANTO TECHNOLOGY LLC (US) 2016-10-06 WO disclosed