SCHEMBL18124148

SCHEMBL18124148

Cc1cc(C(=O)O)ccc1-n1c(CCC(=O)O)ccc1-c1ccc(-c2nn[nH]n2)cc1.Cc1cc(C(N)=O)ccc1-n1c(CCC(=O)O)ccc1-c1ccc(N2CCOCC2)cc1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADH5 P11766 1/20 0.56
CYP2C19 P33261 1/20 0.56
NPC1 O15118 1/20 0.44
POLB P06746 5/20 0.40
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
MAPT P10636 5/20 0.38
TP53 P04637 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 1/20 0.37
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL245380 0.89 ADH5 (0.64) ADH5CYP2C19NPC1POLBMEN1
SCHEMBL244683 0.89 ADH5 (0.67) ADH5CYP2C19NPC1POLBMEN1
SCHEMBL244264 0.87 ADH5 (0.54) ADH5CYP2C19NPC1POLBMEN1
SCHEMBL247303 0.82 ADH5 (0.69) ADH5CYP2C19NPC1POLBMEN1
SCHEMBL244681 0.81 ADH5 (0.66) ADH5CYP2C19NPC1POLBMEN1
SCHEMBL242471 0.81 ADH5 (0.68) ADH5CYP2C19NPC1POLBMEN1
SCHEMBL1834591 0.79 ADH5 (0.52) ADH5CYP2C19POLBMEN1KMT2A
SCHEMBL245660 0.79 ADH5 (0.71) ADH5CYP2C19NPC1POLBMEN1
SCHEMBL244176 0.77 ADH5 (0.74) ADH5CYP2C19NPC1POLBMEN1
SCHEMBL246524 0.76 ADH5 (0.63) ADH5CYP2C19NPC1POLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2318006-B1 NOVEL PYRROLE INHIBITORS OF S-NITROSOGLUTATHIONE REDUCTASE AS THERAPEUTIC AGENTS NIVALIS THERAPEUTICS INC (US) 2016-10-12 EP claimed