SCHEMBL18133045

SCHEMBL18133045

NN1CCC(c2nnc(-c3ccc(F)cc3)o2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.51
CA2 P00918 3/20 0.51
ALDH1A1 P00352 2/20 0.50
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
GRM5 P41594 1/20 0.50
ALOX15B O15296 1/20 0.50
CHRNA7 P36544 2/20 0.48
CYP2C19 P33261 1/20 0.48
MAPT P10636 2/20 0.46
ATM Q13315 1/20 0.45
TNKS O95271 3/20 0.44
PARP1 P09874 2/20 0.44
PARP2 Q9UGN5 1/20 0.44
TSHR P16473 2/20 0.44
POLB P06746 2/20 0.44
TP53 P04637 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
USP2 O75604 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12049758 0.87 GRM5 (0.54) CA1CA2ALDH1A1NPC1RAB9A
SCHEMBL16989766 0.82 CA1 (0.57) CA1CA2ALDH1A1NPC1RAB9A
SCHEMBL16989767 0.82 CA1 (0.57) CA1CA2ALDH1A1NPC1RAB9A
SCHEMBL12026462 0.82 HTR4 (0.54) CA1CA2ALDH1A1NPC1RAB9A
SCHEMBL14637530 0.81 MAPT (0.55) CA1CA2ALDH1A1NPC1RAB9A
SCHEMBL2247489 0.79 NPC1 (0.53) CA1CA2ALDH1A1NPC1RAB9A
SCHEMBL14637620 0.78 TNKS (0.54) CA1CA2ALDH1A1NPC1RAB9A
SCHEMBL16825830 0.77 GRM5 (0.44) CA1CA2ALDH1A1NPC1RAB9A
SCHEMBL27968848 0.76 MAPT (0.50) CA1CA2ALDH1A1GRM5ALOX15B
SCHEMBL21939281 0.75 LRRK2 (0.57) CA1CA2ALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2788086-B1 SUBSTITUTED PYRAZOLES AS MGLU5 RECEPTOR MODULATORS BOEHRINGER INGELHEIM INT (DE) 2016-10-12 EP disclosed